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Article Dans Une Revue SYNLETT Année : 2018

Weinreb β-Ketoamides in Enantioselective Organocatalysis: A Balance between Reactivity and Selectivity

Résumé

β-Dicarbonyl compounds have established themselves as substrates of choice in enantioselective organocatalysis because of their easy activation. Among them, β-diketones, β-diesters and β-ketoesters lead the dance and there has been only limited work with other β-dicarbonyl compounds as pronucleophiles. In this Synpacts article, we wish to discuss our recent contributions to the introduction of Weinreb β-ketoamides in organocatalyzed transformations, where they can provide an interesting balance between reactivity and selectivity, with also interesting potentialities in terms of post-functionalization.
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Dates et versions

hal-01723120 , version 1 (05-03-2018)

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Haiying Du, Yohan Dudognon, Jean Rodriguez, Thierry Constantieux, Xavier Bugaut. Weinreb β-Ketoamides in Enantioselective Organocatalysis: A Balance between Reactivity and Selectivity. SYNLETT, In press, ⟨10.1055/s-0036-1591870⟩. ⟨hal-01723120⟩

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