@article{poras:hal-03292709, TITLE = {{Modulation of disulfide dual ENKephalinase inhibitors (DENKIs) activity by a transient N-protection for pain alleviation by oral route}}, AUTHOR = {Poras, Herve and Bonnard, Elisabeth and Fournie-Zaluski, Marie-Claude and Roques, Bernard P.}, URL = {https://hal-cnrs.archives-ouvertes.fr/hal-03292709}, JOURNAL = {{European Journal of Medicinal Chemistry}}, PUBLISHER = {{Elsevier}}, VOLUME = {102}, PAGES = {58-67}, YEAR = {2015}, DOI = {10.1016/j.ejmech.2015.07.027}, KEYWORDS = {AMINOMETHYL)-1-CYCLOHEXANE ACETIC-ACID ; SCIATIC-NERVE INJURY ; DEGRADING ENZYMES ; GABAPENTIN PRODRUG ; NEUROPATHIC PAIN ; POTENT ; RAT ; HYPERALGESIA ; NOCICEPTION ; ANALGESICS}, HAL_ID = {hal-03292709}, HAL_VERSION = {v1}, }