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authFullName_s : Dirk Tourwé

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

Emilie Eiselt , Simon Gonzalez , Charlotte Martin , Magali Chartier , Cecilia Betti et al.
ACS Chemical Neuroscience, 2019, 10 (11), pp.4535-4544. ⟨10.1021/acschemneuro.9b00390⟩
Journal articles hal-02400886v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors

Jolien de Neve , Thomas M A Barlow , Dirk Tourwé , Frédéric Bihel , Frédéric Simonin et al.
RSC Medicinal Chemistry, 2021
Journal articles hal-03435229v1

Novel, potent and selective angiotensin IV short analogues.

Aneta Lukaszuk , Heidi Demaegdt , Philippe Karoyan , Patrick Vanderheyden , Georges Vauquelin et al.
Journal Of Peptide Science 2008, 2007, 14 ((8)), pp.143-144
Journal articles hal-00423314v1
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Bifunctional Peptide-Based Opioid Agonist–Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic Pain

Karel Guillemyn , Joanna Starnowska , Camille Lagard , Jolanta Dyniewicz , Ewelina Rojewska et al.
Journal of Medicinal Chemistry, 2016, 59 (8), pp.3777-3792. ⟨10.1021/acs.jmedchem.5b01976⟩
Journal articles hal-02993685v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors

Jolien de Neve , Thomas M. A. Barlow , Dirk Tourwé , Frédéric Bihel , Frédéric Simonin et al.
RSC Medicinal Chemistry, 2021, 12 (6), pp.828-870. ⟨10.1039/D1MD00041A⟩
Journal articles hal-03442028v1

#-Homo-amino Acid Scan of Angiotensin IV

Aneta Lukaszuk , Heidi Demaegdt , Erzsebet Szemenyei , Géza Tóth , Dagmara Tymecka et al.
Journal of Medicinal Chemistry, 2008, 51 ((7)), pp.2291-2296 •
Journal articles hal-00423876v1

Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds

Olivier van Der Poorten , Baptiste Legrand , Lubomir Vezenkov , Júlia García-Pindado , Nadir Bettache et al.
ChemBioChem, 2018, 19 (7), pp.696-705. ⟨10.1002/cbic.201700678⟩
Journal articles hal-03564881v1

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds

Olivier van Der Poorten , Robin van den Hauwe , Emilie Eiselt , Cecilia Betti , Karel Guillemyn et al.
ACS Medicinal Chemistry Letters, 2017, 8 (11), pp.1177-1182. ⟨10.1021/acsmedchemlett.7b00347⟩
Journal articles hal-02368778v1

Peptides 1998, Proceedings of the 25th European Peptide Symposium

Joseph Richard Casimir , Marie-Claude Biémont-Trescol , Dirk Tourwé , Joëlle Paris , Laurent Ettouati et al.
B. Sandor and H. Ferenc. 25th European Peptide Symposium, Aug 1998, Budapest, Hungary. Akademiai Kiado, pp.654-655, 1999
Proceedings hal-01709948v1

Indoloazepinone-Containing Oligomers as Cell-Penetrating (Non)Peptides: Synthesis, Structuration and Internalization

Olivier van Der Poorten , Baptiste Legrand , Lubomir Vezenkov , Jean Martinez , Nadir Bettache et al.
Journal of Peptide Science, 2018, 22 (S2), pp.S117. ⟨10.1002/psc.2950⟩
Journal articles hal-03576982v1