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Intestinal Epithelial AMPK Deficiency Causes Delayed Colonic Epithelial Repair in DSS-Induced Colitis
Séverine Olivier
,
Hanna Diounou
,
Camille Pochard
,
Lisa Frechin
,
Emilie Durieu
et al.
Journal articles
hal-03864685v1
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A Collection of Bioactive Nitrogen-Containing Molecules from the Marine Sponge Acanthostrongylophora ingens
Germana Esposito
,
Linh Mai
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Arlette Longeon
,
Alfonso Mangoni
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Emilie Durieu
et al.
Journal articles
hal-02396669v1
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Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell Effects
Solene Guiheneuf
,
Ludovic Paquin
,
Francois Carreaux
,
Emilie Durieu
,
Helene Benedetti
et al.
Journal articles
hal-01114583v1
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Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.
Tania Tahtouh
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Jonathan M. Elkins
,
Panagis Filippakopoulos
,
Meera Soundararajan
,
Guillaume Burgy
et al.
Journal articles
hal-00870472v1
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Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives.
Francis Giraud
,
Georges Alves
,
Eric Debiton
,
Lionel Nauton
,
Vincent Thery
et al.
Journal of Medicinal Chemistry, 2011, 54, pp.4474-4489
Journal articles
hal-00609607v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
,
Eric Goffin
,
Sebastien Dilly
,
Julien Hanson
,
Lionel Pochet
et al.
Journal articles
hal-02141338v1
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An efficient approach to dispacamide A and its derivatives.
Solène Guihéneuf
,
Ludovic Paquin
,
François Carreaux
,
Emilie Durieu
,
Laurent Meijer
et al.
Journal articles
hal-00870469v1
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Synthesis of N,N'-bis(5-arylidene-4-oxo-3,5-dihydro-4H-imidazol-2-yl)diamines bearing various linkers and biological evaluation as potential inhibitors of kinases.
Wacothon Karime Coulibaly
,
Ludovic Paquin
,
Anoubilé Bénie
,
Yves-Alain Bekro
,
Emilie Durieu
et al.
Journal articles
istex
hal-00813182v1
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
Nadège Loaëc
,
Eletta Attanasio
,
Benoît Villiers
,
Emilie Durieu
,
Tania Tahtouh
et al.
Journal articles
hal-01640115v1
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Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors
Tania Tahtouh
,
Emilie Durieu
,
Benoit Villiers
,
Celine Bruyere
,
Thu Lan Nguyen
et al.
Journal articles
hal-03512536v1
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Intestinal Epithelial AMPK Deficiency Causes Delayed Colonic Epithelial Repair in DSS-Induced Colitis
Séverine Olivier
,
Hanna Diounou
,
Camille Pochard
,
Lisa Frechin
,
Emilie Durieu
et al.
Journal articles
inserm-03572820v1
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cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.
Xavier Fant
,
Emilie Durieu
,
Gaëtan Chicanne
,
Bernard Payrastre
,
Diego Sbrissa
et al.
Journal articles
inserm-01012086v1
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Characterisation of tau in the human and rodent enteric nervous system under physiological conditions and in tauopathy
Arthur Lionnet
,
Matthew Wade
,
Anne-Gaëlle Corbillé
,
Alice Prigent
,
Sébastien Paillusson
et al.
Journal articles
hal-03153572v1
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From drug screening to target deconvolution: A target-based drug discovery pipeline using Leishmania casein kinase 1 isoform 2 to identify compounds with anti-leishmanial activity
Emilie Durieu
,
Eric Prina
,
Olivier Leclercq
,
Nassima Oumata
,
Nicolas Gaboriaud-Kolar
et al.
Journal articles
hal-01299756v1
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Chemical synthesis and biological validation of immobilized protein kinase inhibitory Leucettines.
Guillaume Burgy
,
Tania Tahtouh
,
Emilie Durieu
,
Béatrice Foll-Josselin
,
Emmanuelle Limanton
et al.
Journal articles
hal-00822733v1
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Exploring the Synthesis of New 1-(4-Substitutedphenylamino) imidazo[1,5-a]indol-3-one Derivatives as Cyclized Analogs of Leucettines
Guillaume Burgy
,
Emmanuelle Limanton
,
François Carreaux
,
Emilie Durieu
,
Laurent Meijer
et al.
Journal articles
hal-01116022v1
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New 5-ylidene rhodanine derivatives based on the dispacamide A model.
Solène Guihéneuf
,
Ludovic Paquin
,
François Carreaux
,
Emilie Durieu
,
Thierry Roisnel
et al.
Journal articles
hal-01017003v1
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Role of intestinal epithelial AMPK in the protective effect of metformin on dextran sodium sulfate‐induced colitis in mice
Hanna Diounou
,
Severine Olivier
,
Emilie Durieu
,
Marc Foretz
,
Michel Neunlist
et al.
Journal articles
hal-03441649v1
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Pharmacological assessment defines Leishmania donovani casein kinase 1 as a drug target and reveals important functions in parasite viability and intracellular infection
Najma Rachidi
,
Jean François Taly
,
Emilie Durieu
,
Olivier Leclercq
,
Nathalie Aulner
et al.
Journal articles
pasteur-01433412v1
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Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A
Khadidja Bourahla
,
Solène Guihéneuf
,
Emmanuelle Limanton
,
Ludovic Paquin
,
Rémy Le Guével
et al.
Journal articles
hal-03467664v1
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