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authFullName_s : Emilie Durieu
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Intestinal Epithelial AMPK Deficiency Causes Delayed Colonic Epithelial Repair in DSS-Induced Colitis

Séverine Olivier , Hanna Diounou , Camille Pochard , Lisa Frechin , Emilie Durieu et al.
Cells, 2022, 11 (4), pp.590. ⟨10.3390/cells11040590⟩
Journal articles hal-03864685v1

A Collection of Bioactive Nitrogen-Containing Molecules from the Marine Sponge Acanthostrongylophora ingens

Germana Esposito , Linh Mai , Arlette Longeon , Alfonso Mangoni , Emilie Durieu et al.
Marine drugs, 2019, 17 (8), pp.472. ⟨10.3390/md17080472⟩
Journal articles hal-02396669v1

Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell Effects

Solene Guiheneuf , Ludovic Paquin , Francois Carreaux , Emilie Durieu , Helene Benedetti et al.
Current microwave chemistry, 2014, 1 (1), pp.33-40. ⟨10.2174/22133356114019990002⟩
Journal articles hal-01114583v1

Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.

Tania Tahtouh , Jonathan M. Elkins , Panagis Filippakopoulos , Meera Soundararajan , Guillaume Burgy et al.
Journal of Medicinal Chemistry, 2012, 55 (21), pp.9312-30. ⟨10.1021/jm301034u⟩
Journal articles hal-00870472v1

Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives.

Francis Giraud , Georges Alves , Eric Debiton , Lionel Nauton , Vincent Thery et al.
Journal of Medicinal Chemistry, 2011, 54, pp.4474-4489
Journal articles hal-00609607v1
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30th Franco-Belgian conference of pharmacochemistry

Charlotte Bouckaert , Eric Goffin , Sebastien Dilly , Julien Hanson , Lionel Pochet et al.
Pharmaceuticals, 2016, 9 (4), pp.73. ⟨10.3390/ph9040073⟩
Journal articles hal-02141338v1

An efficient approach to dispacamide A and its derivatives.

Solène Guihéneuf , Ludovic Paquin , François Carreaux , Emilie Durieu , Laurent Meijer et al.
Organic & Biomolecular Chemistry, 2012, 10 (5), pp.978-87. ⟨10.1039/c1ob06161e⟩
Journal articles hal-00870469v1

Synthesis of N,N'-bis(5-arylidene-4-oxo-3,5-dihydro-4H-imidazol-2-yl)diamines bearing various linkers and biological evaluation as potential inhibitors of kinases.

Wacothon Karime Coulibaly , Ludovic Paquin , Anoubilé Bénie , Yves-Alain Bekro , Emilie Durieu et al.
European Journal of Medicinal Chemistry, 2012, 58, pp.581-90. ⟨10.1016/j.ejmech.2012.08.044⟩
Journal articles istex hal-00813182v1
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases

Nadège Loaëc , Eletta Attanasio , Benoît Villiers , Emilie Durieu , Tania Tahtouh et al.
Marine drugs, 2017, 15 (10), pp.316 -. ⟨10.3390/md15100316⟩
Journal articles hal-01640115v1

Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors

Tania Tahtouh , Emilie Durieu , Benoit Villiers , Celine Bruyere , Thu Lan Nguyen et al.
Journal of Medicinal Chemistry, 2022, 65 (2), pp.1396-1417. ⟨10.1021/acs.jmedchem.1c01141⟩
Journal articles hal-03512536v1
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Intestinal Epithelial AMPK Deficiency Causes Delayed Colonic Epithelial Repair in DSS-Induced Colitis

Séverine Olivier , Hanna Diounou , Camille Pochard , Lisa Frechin , Emilie Durieu et al.
Cells, 2022, 11 (4), pp.590. ⟨10.3390/cells11040590⟩
Journal articles inserm-03572820v1

cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.

Xavier Fant , Emilie Durieu , Gaëtan Chicanne , Bernard Payrastre , Diego Sbrissa et al.
Molecular Pharmacology, 2014, 85 (3), pp.441-50. ⟨10.1124/mol.113.090837⟩
Journal articles inserm-01012086v1
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Characterisation of tau in the human and rodent enteric nervous system under physiological conditions and in tauopathy

Arthur Lionnet , Matthew Wade , Anne-Gaëlle Corbillé , Alice Prigent , Sébastien Paillusson et al.
Acta Neuropathologica Communications, 2018, 6 (1), ⟨10.1186/s40478-018-0568-3⟩
Journal articles hal-03153572v1
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From drug screening to target deconvolution: A target-based drug discovery pipeline using Leishmania casein kinase 1 isoform 2 to identify compounds with anti-leishmanial activity

Emilie Durieu , Eric Prina , Olivier Leclercq , Nassima Oumata , Nicolas Gaboriaud-Kolar et al.
Antimicrobial Agents and Chemotherapy, 2016, ⟨10.1128/AAC.00021-16⟩
Journal articles hal-01299756v1

Chemical synthesis and biological validation of immobilized protein kinase inhibitory Leucettines.

Guillaume Burgy , Tania Tahtouh , Emilie Durieu , Béatrice Foll-Josselin , Emmanuelle Limanton et al.
European Journal of Medicinal Chemistry, 2013, 62, pp.728-37. ⟨10.1016/j.ejmech.2013.01.035⟩
Journal articles hal-00822733v1
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Exploring the Synthesis of New 1-(4-Substitutedphenylamino) imidazo[1,5-a]indol-3-one Derivatives as Cyclized Analogs of Leucettines

Guillaume Burgy , Emmanuelle Limanton , François Carreaux , Emilie Durieu , Laurent Meijer et al.
Journal of Applied Pharmaceutical Science, 2014, 4 (6), pp.25 - 32. ⟨10.7324/JAPS.2014.40604⟩
Journal articles hal-01116022v1
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New 5-ylidene rhodanine derivatives based on the dispacamide A model.

Solène Guihéneuf , Ludovic Paquin , François Carreaux , Emilie Durieu , Thierry Roisnel et al.
Molecular Diversity, 2014, 18 (2), pp.375-88. ⟨10.1007/s11030-014-9509-7⟩
Journal articles hal-01017003v1

Role of intestinal epithelial AMPK in the protective effect of metformin on dextran sodium sulfate‐induced colitis in mice

Hanna Diounou , Severine Olivier , Emilie Durieu , Marc Foretz , Michel Neunlist et al.
FASEB Journal, 2021, 35 (S1), ⟨10.1096/fasebj.2021.35.S1.03621⟩
Journal articles hal-03441649v1

Pharmacological assessment defines Leishmania donovani casein kinase 1 as a drug target and reveals important functions in parasite viability and intracellular infection

Najma Rachidi , Jean François Taly , Emilie Durieu , Olivier Leclercq , Nathalie Aulner et al.
Antimicrobial Agents and Chemotherapy, 2014, 58 (3), pp.1501-1515. ⟨10.1128/AAC.02022-13⟩
Journal articles pasteur-01433412v1
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Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A

Khadidja Bourahla , Solène Guihéneuf , Emmanuelle Limanton , Ludovic Paquin , Rémy Le Guével et al.
Pharmaceuticals, 2021, 14 (11), pp.1086-1117. ⟨10.3390/ph14111086⟩
Journal articles hal-03467664v1