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Substituted thiazolamide coupled to a redox delivery system: a new γ-secretase inhibitor with enhanced pharmacokinetic profile
Younes Laras
,
Gilles Quéléver
,
Cédrik Garino
,
Nicolas Pietrancosta
,
Mahmoud Sheha
et al.
Journal articles
istex
hal-02351730v1
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Development of a L-Tryptophan-Based Ligand for Regioselective Copper Catalyzed N 2 -Arylation of 1,2,3-Triazoles
Alexandra Basilio Lopes
,
Patrick Wagner
,
Arthur Eugen Kümmerle
,
Frédéric Bihel
,
Jean-Jacques Bourguignon
et al.
Journal articles
hal-02368798v1
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Development of a Peptidomimetic Antagonist of Neuropeptide FF Receptors for the Prevention of Opioid-Induced Hyperalgesia
Frédéric Bihel
,
Jean-Paul Humbert
,
Severine Schneider
,
Isabelle Bertin
,
Patrick Wagner
et al.
Journal articles
hal-03198603v1
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Erratum to: "CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors
Saleh Mones
,
Burkhard Gess
,
Benoit Bordignon
,
Alexandre Altie
,
Peter Young
et al.
Journal articles
hal-02630248v1
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Microwave-assisted cyclic amidine synthesis using TiCl4
Hellal Malik
,
Frédéric Bihel
,
Bourguignon Jean-Jacques
Journée Scientifique de l'IFR Gilbert Laustriat, 2006, Illkirch, France
Conference papers
hal-00195376v1
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Human erythrocytes release ATP by a novel pathway involving VDAC oligomerization independent of pannexin-1
Irene Marginedas-Freixa
,
Cora Lilia Alvarez
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Martina Moras
,
María Florencia Leal Denis
,
Claude Hattab
et al.
Journal articles
hal-02368694v1
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A bifunctional-biased mu-opioid agonist–neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects
Armand Drieu La Rochelle
,
Karel Guillemyn
,
Maria Dumitrascuta
,
Charlotte Martin
,
Valérie Utard
et al.
Journal articles
hal-02368742v1
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6-Endo-dig cyclization of heteroarylesters to alkynes promoted by Lewis acid catalyst in presence of Brønsted acid
Frédéric Bihel
,
Hellal Malik
,
Bourguignon Jean-Jacques
XXVII REGIO, Sep 2007, Buhl, France
Conference papers
hal-00195398v1
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Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new β-amyloid peptide production inhibitors and their activities on various classes of protease
Agnès Petit-Paitel
,
Frédéric Bihel
,
Gilles Quéléver
,
Hugues Lelouard
,
Agnès Petit
et al.
Journal articles
istex
hal-03016636v1
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Mitochondria modulatory effects of new TSPO ligands in a cellular model of tauopathies
Amandine Grimm
,
Imane Lejri
,
François Hallé
,
Martine Schmitt
,
Jürgen Götz
et al.
Journal articles
hal-02368671v1
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Development of Dipeptidic hGPR54 Agonists
Christelle Doebelin
,
Isabelle I. Bertin
,
Séverine Schneider
,
Martine Schmitt
,
Jean-Jacques Bourguignon
et al.
Journal articles
istex
hal-02368845v1
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RF-amide neuropeptides and their receptors in Mammals: Pharmacological properties, drug development and main physiological functions
Raphaelle Quillet
,
Safia Ayachi
,
Frédéric Bihel
,
Khadija Elhabazi
,
Brigitte Ilien
et al.
Journal articles
hal-02368835v1
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New b-strand macrocyclic peptidomimetic analogues containing alpha-(O-, S- or NH-)aryl substituted glycine residues: synthesis, chemical and enzymatic properties
Gilles Quéléver
,
Frédéric Bihel
,
Jean-Louis Kraus
Organic & Biomolecular Chemistry, 2003, 1, pp.1676-1683
Journal articles
hal-00154124v1
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6-Endo-dig cyclization of heteroarylesters to alkynes promoted by Lewis acid catalyst in presence of Brønsted acid
Hellal Malik
,
Bourguignon Jean-Jacques
,
Frédéric Bihel
SAJEC, Oct 2007, Paris, France
Conference papers
hal-00195387v1
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Diastereoselective Synthesis of Nonplanar 3-Amino-1,2,4-oxadiazine Scaffold: Structure Revision of Alchornedine
Shuang-Qi Tang
,
Maeva Leloire
,
Severine Schneider
,
Julie Mohr
,
Jacques Bricard
et al.
Journal articles
hal-03021041v1
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Opioid adjuvant strategy: improving opioid effectiveness
Frédéric Bihel
Journal articles
hal-02368859v1
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Discovery of Imidazoquinazolinone Derivatives as TSPO Ligands Modulating Neurosteroidogenesis and Cellular Bioenergetics in Neuroblastoma Cells Expressing Amyloid Precursor Protein
François Hallé
,
Imane Lejri
,
Mustapha Abarghaz
,
Amandine Grimm
,
Christian Klein
et al.
Journal articles
hal-02368811v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
Jolien de Neve
,
Thomas M. A. Barlow
,
Dirk Tourwé
,
Frédéric Bihel
,
Frédéric Simonin
et al.
Journal articles
hal-03442028v1
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The translocator protein ligand XBD173 improves clinical symptoms and neuropathological markers in the SJL/J mouse model of multiple sclerosis
I. Marginedas-Freixa
,
C. Hattab
,
G. Bouyer
,
F. Halle
,
A. Chene
et al.
Journal articles
hal-02290250v1
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Synthesis of 3-amino-3,4-dihydro-1H-quinolin-2-ones through regioselective palladium-catalyzed intramolecular cyclization
François Hallé
,
Olivier van Der Poorten
,
Christelle Doebelin
,
Marie Niederst
,
Séverine Schneider
et al.
Journal articles
hal-02290245v1
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CamKII inhibitors reduce mitotic instability, connexon anomalies and progression of the in vivo behavioral phenotype in transgenic animals expressing a mutated Gjb1 gene
Saleh Mones
,
Benoit Bordignon
,
Franck Peiretti
,
Jean-Francois Landrier
,
Burkhardt Gess
et al.
Journal articles
hal-02639042v1
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6-Endo-dig cyclization of heteroarylesters to alkynes promoted by Lewis acid catalyst in the presence of Bronsted acid
Hellal Malik
,
Bourguignon Jean-Jacques
,
Frédéric Bihel
Tetrahedron Letters, 2008, 49 (1), pp.62-65
Journal articles
hal-00195333v1
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POxAP Precatalysts and the Negishi Cross-Coupling Reaction
Shuang-Qi Tang
,
Martine Schmitt
,
Frédéric Bihel
Journal articles
hal-02997250v1
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Anti-prion Drugs Targeting the Protein Folding Activity of the Ribosome Reduce PABPN1 Aggregation
Aline Bamia
,
Maha Sinane
,
Rima Naït-Saïdi
,
Jamila Dhiab
,
Marc Keruzoré
et al.
Journal articles
hal-03158577v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
Jolien de Neve
,
Thomas M A Barlow
,
Dirk Tourwé
,
Frédéric Bihel
,
Frédéric Simonin
et al.
RSC Medicinal Chemistry, 2021
Journal articles
hal-03435229v1
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Design and synthesis of 3-aminophthalazine derivatives and structural analogues as PDE5 inhibitors: anti-allodynic effect against neuropathic pain in a mouse model
Maud Bollenbach
,
Claire Lugnier
,
M Elanie Kremer
,
Eric Salvat
,
Salim Megat
et al.
Journal articles
hal-02322399v1
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Identification of 8-Hydroxyquinoline Derivatives That Decrease Cystathionine Beta Synthase (CBS) Activity
Pierre Conan
,
Alice Léon
,
Mathilde Gourdel
,
Claire Rollet
,
Loubna Chaïr
et al.
Journal articles
hal-03701324v1
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Efficient and Mild Ullmann-Type N-Arylation of Amides, Carbamates, and Azoles in Water
Maud Bollenbach
,
Pedro Aquino
,
João Xavier De araújo-Júnior
,
Jean-Jacques Bourguignon
,
Frédéric Bihel
et al.
Journal articles
hal-02368823v1
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RF313, an orally bioavailable neuropeptide FF receptor antagonist, opposes effects of RF-amide-related peptide-3 and opioid-induced hyperalgesia in rodents
Khadija Elhabazi
,
Jean-Paul Humbert
,
Isabelle Bertin
,
Raphaelle Quillet
,
Valérie Utard
et al.
Journal articles
hal-01603852v1
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Structure-activity relationship study around guanabenz identifies two derivatives retaining antiprion activity but having lost alpha 2-adrenergic receptor agonistic activity
- Phu Hai Nguyen
,
Hassan Hammoud
,
Sophie Halliez
,
Yanhong Pang
,
Justine Evrard
et al.
Journal articles
hal-02635473v1
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