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authFullName_s : Frédéric Buron

Pyridine-based lanthanide complexes combining MRI and NIR luminescence activities.

Célia S Bonnet , Frédéric Buron , Fabien Caillé , Chad M Shade , Bohuslav Drahoš et al.
Chemistry - A European Journal, 2012, 18 (5), pp.1419-31. ⟨10.1002/chem.201102310⟩
Journal articles istex hal-00720541v1

Development of a bio­active fluorescent inhibitor probe targeting the Rho kinase ROCK for monitoring inhibition action

Justine Corret , Sokaina Hammoud , Frédéric Buron , Pierre Daligaux , Christophe Chesné et al.
FEBS 2021, the 45th FEBS Congress, Jul 2021, Lnubljana, virtual, Slovenia
Conference poster hal-03679980v1
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A Novel Polyaminocarboxylate Compound To Treat Murine Pulmonary Aspergillosis by Interfering with Zinc Metabolism

Paris Laskaris , Rocío Vicentefranqueira , Olivier Helynck , Grégory Jouvion , José Antonio Calera et al.
Antimicrobial Agents and Chemotherapy, 2018, 62 (6), pp.e02510-17. ⟨10.1128/AAC.02510-17⟩
Journal articles pasteur-01968421v1

Analytical developments for 47 pesticides: first identification of neutral chloroacetanilide derivatives in French groundwater

Laurence Amalric , Nicole Baran , Charlotte Coureau , Lucie Maingot , Frédéric Buron et al.
International Journal of Environmental Analytical Chemistry, 2013, 93 (15), pp.1660-1675. ⟨10.1080/03067319.2013.853758⟩
Journal articles hal-00975875v1

Synthesis of chromeno[3,4-b]indoles as Lamellarin D analogues: a novel DYRK1A inhibitor class.

Cleopatra Neagoie , Emeline Vedrenne , Frédéric Buron , Jean-Yves Mérour , Sorin Rosca et al.
European Journal of Medicinal Chemistry, 2012, 49, pp.379-96. ⟨10.1016/j.ejmech.2012.01.040⟩
Journal articles istex hal-00726237v1

Lanthanide-Based, Near-Infrared Luminescent and Magnetic Lipoparticles: Monitoring Particle Integrity.

Sara Lacerda , Célia S Bonnet , Agnès Pallier , Sandrine Villette , Frédéric Foucher et al.
Small, 2013, 9 (16), pp.2662-2666. ⟨10.1002/smll.201201923⟩
Journal articles istex hal-00817465v1

Hydrophobic chromophore cargo in micellar structures: a different strategy to sensitize lanthanide cations

Célia Bonnet , Laurent Pellegatti , Frédéric Buron , Chad Shade , Sandrine Villette et al.
Chemical Communications, 2010, 46 (1), pp.124-126. ⟨10.1039/B918881A⟩
Journal articles istex hal-02117713v1
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Design, Synthesis and SAR in 2,4,7-Trisubstituted Pyrido[3,2-d]Pyrimidine Series as Novel PI3K/mTOR Inhibitors

Frédéric Buron , Nuno Rodrigues , Thibault Saurat , Marie-Aude Hiebel , Stéphane Bourg et al.
Molecules, 2021, 26 (17), pp.5349. ⟨10.3390/molecules26175349⟩
Journal articles hal-03348966v1

Synthesis of γ-carboline N-oxide under gold(I)-catalysis and C-1 amino and fluoro γ-carboline

Zak Agnieszka , Hamid Marzag , Rodrigues Nuno , Vercouillie Johnny , Sylvie Chalon et al.
Tetrahedron, 2021, 89, pp.132154. ⟨10.1016/j.tet.2021.132154⟩
Journal articles hal-03717446v1
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Development and preclinical evaluation of [18F]FBVM as a new potent PET tracer for vesicular acetylcholine transporter

Johnny Vercouillie , Frédéric Buron , Sophie Sérrière , Nuno Rodrigues , Zuhal Gulhan et al.
European Journal of Medicinal Chemistry, 2022, 244, pp.114794. ⟨10.1016/j.ejmech.2022.114794⟩
Journal articles hal-03881143v1
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Design and biological evaluation of substituted 5,7-dihydro-6 H -indolo[2,3- c ]quinolin-6-one as novel selective Haspin inhibitors

Sreenivas Avula , Xudan Peng , Xingfen Lang , Micky Tortorella , Béatrice Josselin et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2022, 37 (1), pp.1632-1650. ⟨10.1080/14756366.2022.2082419⟩
Journal articles hal-03818922v1

Selection of Bis-Indolyl Pyridines and Triphenylamines as New Inhibitors of SARS-CoV-2 Cellular Entry by Modulating the Spike Protein/ACE2 Interfaces

Delphine Lapaillerie , Cathy Charlier , Véronique Guyonnet-Dupérat , Emilie Murigneux , Henrique Fernandes et al.
Antimicrobial Agents and Chemotherapy, 2022, 66 (8), ⟨10.1128/aac.00083-22⟩
Journal articles hal-03821963v1

Development of a bio­active fluorescent inhibitor probe targeting the Rho kinase ROCK for monitoring inhibition action

Justine Corret , Sokaina Hammoud , Frédéric Buron , Pierre Daligaux , Christophe Chesné et al.
FEBS 2021, the 45th FEBS Congress, Jul 2021, Virtual, France
Conference papers hal-03668584v1

Modeling Temperature and Species Concentration Profiles on a Continuous-Flow Reactor Applied to Aldol Condensation

Aziza Chairat , Mazarine Laurent , Sylvain Routier , Frédéric Buron , Stephane Bostyn et al.
ACS Omega, 2022, 7 (23), pp.19166-19175. ⟨10.1021/acsomega.2c00079⟩
Journal articles hal-03705725v1
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Glycosaminoglycan mimetics obtained by microwave-assisted sulfation of marine bacterium sourced infernan exopolysaccharide

Sylvia Colliec-Jouault , Fabiana Esposito , Hélène Ledru , Corinne Sinquin , Arnaud Fillaudeau et al.
Biomacromolecules, 2023, 24, pp.462-470. ⟨10.1021/acs.biomac.2c01277⟩
Journal articles hal-03948691v1
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3

Killian Oukoloff , Nicolas Coquelle , Manuela Bartolini , Marina Naldi , Rémy Le Guével et al.
European Journal of Medicinal Chemistry, 2019, 168, pp.58-77. ⟨10.1016/j.ejmech.2018.12.063⟩
Journal articles hal-02055769v1

PiB-Conjugated, Metal-Based Imaging Probes: Multimodal Approaches for the Visualization of β-Amyloid Plaques

André Martins , Jean-François Morfin , Anna Kubíčková , Vojtěch Kubíček , Frédéric Buron et al.
ACS Medicinal Chemistry Letters, 2013, 4 (5), pp.436-440. ⟨10.1021/ml400042w⟩
Journal articles hal-03572643v1

Towards a biomimetic synthesis of barrenazine A

Frédéric Buron , Alain Turck , Nelly Plé , Laurent Bischoff , Francis Marsais et al.
Tetrahedron Letters, 2007, 48 (25), pp.4327-4330. ⟨10.1016/j.tetlet.2007.04.108⟩
Journal articles istex hal-02385028v1

Isoquinoline-based lanthanide complexes: bright NIR optical probes and efficient MRI agents.

Fabien Caillé , Célia S Bonnet , Frédéric Buron , Sandrine Villette , Lothar Helm et al.
Inorganic Chemistry, 2012, 51 (4), pp.2522-32. ⟨10.1021/ic202446e⟩
Journal articles hal-00721803v1

PiB-Conjugated, Metal-Based Imaging Probes: Multimodal Approaches for the Visualization of β-Amyloid Plaques

André F. Martins , Jean-François Morfin , Anna Kubícková , Vojtěch Kubícek , Frédéric Buron et al.
Planetary and Space Science, 2013, 4 (5), pp.436-440. ⟨10.1021/ml400042w⟩
Journal articles hal-00840181v1

Synthesis and biological evaluation of 2,3-bis(het)aryl-4-azaindole derivatives as protein kinase inhibitors

Frédéric Pin , Frédéric Buron , Fabienne Saab , Lionel Colliandre , Stéphane Bourg et al.
MedChemComm, 2011, 2 (9), pp.899-903. ⟨10.1039/c1md00141h⟩
Journal articles hal-00720699v1
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New in-capillary electrophoretic kinase assays to evaluate inhibitors of the PI3k/Akt/mTOR signaling pathway

Reine Nehmé , Hala Nehmé , Thibault Saurat , Marie-Ludivine De-Tauzia , Frédéric Buron et al.
Analytical and Bioanalytical Chemistry, 2014, 406 (15), pp.3743-3754. ⟨10.1007/s00216-014-7790-z⟩
Journal articles hal-01180770v1

On the racemisation of aspartic anhydride during its preparation

Frédéric Buron , Geoffrey Deguest , Laurent Bischoff , Corinne Fruit , Francis Marsais et al.
Tetrahedron: Asymmetry, 2007, 18 (13), pp.1625-1627. ⟨10.1016/j.tetasy.2007.07.003⟩
Journal articles istex hal-02385023v1

Screening of Activation Tools to Design Sulfated Saccharides

Hélène Ledru , Joseph d'Attoma , Stéphane Bostyn , Sylvain Routier , Frédéric Buron et al.
ChemistrySelect, 2017, 2 (30), pp.9637-9641. ⟨10.1002/slct.201701853⟩
Journal articles hal-03283191v1
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A facile one-pot synthesis of new poly functionalized pyrrolotriazoles via a regioselective multicomponent cyclisation and Suzuki–Miyaura coupling reactions

Simon Garnier , Kévin Brugemann , Agnieszka Zak , Johnny Vercouillie , Marie Potier-Cartereau et al.
Catalysts, 2022, 12 (8), pp.828. ⟨10.3390/catal12080828⟩
Journal articles hal-03820676v1
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Design of new disubstituted imidazo[1,2- b ]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation

Jonathan Elie , Omid Feizbakhsh , Nathalie Desban , Béatrice Josselin , Blandine Baratte et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2020, 35 (1), pp.1840-1853. ⟨10.1080/14756366.2020.1825408⟩
Journal articles hal-03004407v1

Design, Synthesis, and Biological Activity of Pyridopyrimidine Scaffolds as Novel PI3K/mTOR Dual Inhibitors

Thibault Saurat , Frédéric Buron , Nuno Rodrigues , Marie-Ludivine de Tauzia , Lionel Colliandre et al.
Journal of Medicinal Chemistry, 2014, 57 (3), pp.613-631. ⟨10.1021/jm401138v⟩
Journal articles hal-01180887v1

A pyridine-based ligand with two hydrazine functions for lanthanide chelation: remarkable kinetic inertness for a linear, bishydrated complex

Célia S. Bonnet , Sophie Laine , Frédéric Buron , Gyula Tircsó , Agnès Pallier et al.
Inorganic Chemistry, 2015, 54 (12), pp.5991-6003. ⟨10.1021/acs.inorgchem.5b00804⟩
Journal articles hal-01196977v1
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Selection of Bis-Indolyl Pyridines and Triphenylamines as New Inhibitors of SARS-CoV-2 Cellular Entry by Modulating the Spike Protein/ACE2 Interfaces

Delphine Lapaillerie , Cathy Charlier , Véronique Guyonnet-Dupérat , Emilie Murigneux , Henrique S Fernandes et al.
Antimicrobial Agents and Chemotherapy, 2022, 66 (8), ⟨10.1128/aac.00083-22⟩
Journal articles hal-03826873v1

A Novel Polyaminocarboxylate Compound To Treat Murine Pulmonary Aspergillosis by Interfering with Zinc Metabolism

Paris Laskaris , Rocío Vicentefranqueira , Olivier Helynck , Grégory Jouvion , José Antonio Calera et al.
Antimicrobial Agents and Chemotherapy, 2018, 62 (6), ⟨10.1128/AAC.02510-17⟩
Journal articles hal-03652524v1