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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
Jolien de Neve
,
Thomas M. A. Barlow
,
Dirk Tourwé
,
Frédéric Bihel
,
Frédéric Simonin
et al.
Journal articles
hal-03442028v1
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Characterization of anti-GASP motif antibodies that inhibit the interaction between GPRASP1 and G protein-coupled receptors
Gabrielle Zeder Lutz
,
Olivier Bornert
,
Rosine Fellmann-Clauss
,
Adeline Knittel-Obrecht
,
Thibaud Tranchant
et al.
Journal articles
hal-04029386v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
Jolien de Neve
,
Thomas M A Barlow
,
Dirk Tourwé
,
Frédéric Bihel
,
Frédéric Simonin
et al.
RSC Medicinal Chemistry, 2021
Journal articles
hal-03435229v1
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Behavioral Characterization, Potential Clinical Relevance and Mechanisms of Latent Pain Sensitization
Manon Gerum
,
Frédéric Simonin
Pharmacology & Therapeutics, 2022, 233, pp.108032
Journal articles
hal-03435269v1
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RF9, a potent and selective neuropeptide FF receptor antagonist, prevents opioid-induced tolerance associated with hyperalgesia.
Frédéric Simonin
,
Martine Schmitt
,
Jean-Paul Laulin
,
Emilie Laboureyras
,
Jack H Jhamandas
et al.
Proceedings of the National Academy of Sciences of the United States of America, 2006, 103 (2), pp.466-71. ⟨10.1073/pnas.0502090103⟩
Journal articles
hal-00188146v1
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Morphine-induced hyperalgesia involves mu opioid receptors and the metabolite morphine-3-glucuronide
Laurie-Anne Roeckel
,
Valérie Utard
,
David Reiss
,
Jinane Mouheiche
,
Hervé Maurin
et al.
Journal articles
hal-03448002v1
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A bifunctional-biased mu-opioid agonist–neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects
Armand Drieu La Rochelle
,
Karel Guillemyn
,
Maria Dumitrascuta
,
Charlotte Martin
,
Valérie Utard
et al.
Journal articles
hal-02368742v1
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Development of Dipeptidic hGPR54 Agonists
Christelle Doebelin
,
Isabelle I. Bertin
,
Séverine Schneider
,
Martine Schmitt
,
Jean-Jacques Bourguignon
et al.
Journal articles
istex
hal-02368845v1
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RF-amide neuropeptides and their receptors in Mammals: Pharmacological properties, drug development and main physiological functions
Raphaelle Quillet
,
Safia Ayachi
,
Frédéric Bihel
,
Khadija Elhabazi
,
Brigitte Ilien
et al.
Journal articles
hal-02368835v1
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Attenuated behavioural responses to acute and chronic cocaine in GASP-1-deficient mice
Julien Boeuf
,
José Manuel Trigo
,
Pierre-Henri Moreau
,
Lucas Lecourtier
,
Elise Vogel
et al.
Journal articles
hal-03037839v1
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Recombinant Human Melatonin Receptor MT1 Isolated in Mixed Detergents Shows Pharmacology Similar to That in Mammalian Cell Membranes
Christel Logez
,
Sylvie Berger
,
Céline Legros
,
Jean-Louis Baneres
,
William Cohen
et al.
Journal articles
hal-03573074v1
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Aminoguanidine Hydrazone Derivatives as Nonpeptide NPFF1 Receptor Antagonists Reverse Opioid Induced Hyperalgesia
Hassan Hammoud
,
Khadija Elhabazi
,
Isabelle Bertin
,
Valeŕie Utard
,
Emilie Laboureyras
et al.
Journal articles
hal-02323065v1
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RF313, an orally bioavailable neuropeptide FF receptor antagonist, opposes effects of RF-amide-related peptide-3 and opioid-induced hyperalgesia in rodents
Khadija Elhabazi
,
Jean-Paul Humbert
,
Isabelle Bertin
,
Raphaelle Quillet
,
Valérie Utard
et al.
Journal articles
hal-01603852v1
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Identification of an N -acylated- D Arg-Leu-NH 2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Raphaëlle Quillet
,
Séverine Schneider
,
Valérie Utard
,
Armand Drieu La Rochelle
,
Khadija Elhabazi
et al.
Journal articles
hal-03363456v1
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Behavioral characterization, potential clinical relevance and mechanisms of latent pain sensitization
Manon Gerum
,
Frédéric Simonin
Journal articles
hal-03698407v1
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Disruption of the kappa-opioid receptor gene in mice enhances sensitivity to chemical visceral pain, impairs pharmacological actions of the selective kappa-agonist U-50,488H and attenuates morphine withdrawal
Frédéric Simonin
,
Olga Valverde
,
Claire Smadja
,
Susan Slowe
,
Ian Kitchen
et al.
Journal articles
hal-04017114v1
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