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authFullName_s : Piotr Popik

Novel non-sulfonamide 5-HT 6 receptor partial inverse agonist in a group of imidazo[4,5- b ]pyridines with cognition enhancing properties

David Vanda , Miroslav Soural , Vittorio Canale , Séverine Chaumont-Dubel , Grzegorz Satała et al.
European Journal of Medicinal Chemistry, 2018, 144, pp.716-729. ⟨10.1016/j.ejmech.2017.12.053⟩
Journal articles hal-02366387v1
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Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT 3 and 5-HT 6 Receptor Antagonist with Antipsychotic and Procognitive Properties

Paweł Zajdel , Katarzyna Grychowska , Szczepan Mogilski , Rafał Kurczab , Grzegorz Satała et al.
Journal of Medicinal Chemistry, 2021, 64 (18), pp.13279-13298. ⟨10.1021/acs.jmedchem.1c00224⟩
Journal articles hal-03357806v1
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Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines

Katarzyna Grychowska , Agnieszka Olejarz-Maciej , Klaudia Blicharz , Wojciech Pietruś , Tadeusz Karcz et al.
European Journal of Medicinal Chemistry, 2022, 236, pp.114329. ⟨10.1016/j.ejmech.2022.114329⟩
Journal articles hal-03648220v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity

Marcin Drop , Vittorio Canale , Séverine Chaumont-Dubel , Rafał Kurczab , Grzegorz Satała et al.
ACS Chemical Neuroscience, 2021, 12 (7), pp.1228-1240. ⟨10.1021/acschemneuro.1c00061⟩
Journal articles hal-03192567v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties

Vittorio Canale , Katarzyna Grychowska , Rafał Kurczab , Mateusz Ryng , Abdul Raheem Keeri et al.
European Journal of Medicinal Chemistry, 2020, 208, pp.112765. ⟨10.1016/j.ejmech.2020.112765⟩
Journal articles hal-03029988v1
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Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease

Katarzyna Grychowska , Grzegorz Satala , Tomasz Kos , Anna Partyka , Evelina Colacino et al.
ACS Chemical Neuroscience, 2016, 7 (7), pp.972--83. ⟨10.1021/acschemneuro.6b00090⟩
Journal articles hal-01941175v1
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Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity

Katarzyna Grychowska , Séverine Chaumont-Dubel , Rafał Kurczab , Paulina Koczurkiewicz , Caroline Deville et al.
ACS Chemical Neuroscience, 2019, 10 (7), pp.3183-3196. ⟨10.1021/acschemneuro.8b00618⟩
Journal articles hal-02364291v1