|
|
Novel non-sulfonamide 5-HT 6 receptor partial inverse agonist in a group of imidazo[4,5- b ]pyridines with cognition enhancing properties
David Vanda
,
Miroslav Soural
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Grzegorz Satała
et al.
Journal articles
hal-02366387v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT 3 and 5-HT 6 Receptor Antagonist with Antipsychotic and Procognitive Properties
Paweł Zajdel
,
Katarzyna Grychowska
,
Szczepan Mogilski
,
Rafał Kurczab
,
Grzegorz Satała
et al.
Journal articles
hal-03357806v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines
Katarzyna Grychowska
,
Agnieszka Olejarz-Maciej
,
Klaudia Blicharz
,
Wojciech Pietruś
,
Tadeusz Karcz
et al.
Journal articles
hal-03648220v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity
Marcin Drop
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Grzegorz Satała
et al.
Journal articles
hal-03192567v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
Vittorio Canale
,
Katarzyna Grychowska
,
Rafał Kurczab
,
Mateusz Ryng
,
Abdul Raheem Keeri
et al.
Journal articles
hal-03029988v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease
Katarzyna Grychowska
,
Grzegorz Satala
,
Tomasz Kos
,
Anna Partyka
,
Evelina Colacino
et al.
Journal articles
hal-01941175v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity
Katarzyna Grychowska
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Paulina Koczurkiewicz
,
Caroline Deville
et al.
Journal articles
hal-02364291v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|