Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Bruno Oyallon
,
Marie Brachet-Botineau
,
Cédric Logé
,
Pascal Bonnet
,
Mohamed Souab
et al.
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hal-03408667v1
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A Peak of H3T3 Phosphorylation Occurs in Synchrony with Mitosis in Sea Urchin Early Embryos
Omid Feizbakhsh
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Florian Pontheaux
,
Virginie Glippa
,
Julia Morales
,
Sandrine Ruchaud
et al.
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hal-02536773v1
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The Canadian Prairie Plant Thermopsis rhombifolia Contains Luteolin, a Flavone that Inhibits Cyclin Dependent Kinase 9 and Arrest Cells in the G1-Phase of the Cell Cycle
Jan Tuescher
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Deserae Tailfeathers
,
Sophie Kernéis
,
Blandine Baratte
,
Sandrine Ruchaud
et al.
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hal-03868334v1
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Neurymenolide A, a Novel Mitotic Spindle Poison from the New Caledonian Rhodophyta Phacelocarpus neurymenioides
Sofia-Eléna Motuhi
,
Omid Feizbakhsh
,
Beatrice Foll-Josselin
,
Blandine Baratte
,
Claire Delehouze
et al.
Marine drugs , 2019, Cell Stress, Canonical and Non-Canonical Cell Death Modalities by Marine Natural Compounds and Derivatives, 17 (2), pp.93.
⟨10.3390/md17020093⟩
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hal-02088007v1
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Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration
Viet Hung Dao
,
Isabelle Ourliac-Garnier
,
Marc-Antoine Bazin
,
Catherine Jacquot
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Blandine Baratte
et al.
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hal-03011408v1
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Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition
Hannah Winfield
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Michael Cahill
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Kevin O'Shea
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Larry Pierce
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Thomas Robert
et al.
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hal-03011414v1
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Synthesis and biological evaluation of Haspin inhibitors: kinase inhibitory potency and cellular activity
Wael Zeinyeh
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Yannick Esvan
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Béatrice Josselin
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Mathilde Defois
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Blandine Baratte
et al.
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hal-03764791v1
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Bioprospecting Marine Plankton
Heni Abida
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Sandrine Ruchaud
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Laurent Rios
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Anne Humeau
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Ian Probert
et al.
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hal-01258229v1
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Synthesis and kinase inhibitory potencies of new pyrido[3,4-g]quinazolines substituted at the 8-position
Yannick Esvan
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Béatrice Josselin
,
Blandine Baratte
,
Stéphane Bach
,
Sandrine Ruchaud
et al.
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hal-02926291v1
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
,
Wacothon Karime Coulibaly
,
Yves-Alain Bekro
,
Janat A. Mamyrbekova-Bekro
,
Beatrice Foll-Josselin
et al.
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hal-01414293v1
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High-Throughput Screening of marine resources
Arnaud Hochard
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Luc Reininger
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Sandrine Ruchaud
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Stéphane Bach
Book sections
hal-03871307v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury Halauko
et al.
Journal articles
hal-03875302v1
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New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis
Helmi Tazarki
,
Wael Zeinyeh
,
Yannick J. Esvan
,
Stefan Knapp
,
Deep Chatterjee
et al.
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hal-02150788v1
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Synthesis and evaluation of C3 substituted chalcone‐based derivatives of 7‐azaindole as protein kinase inhibitors
Malikotsi Qhobosheane
,
Lesetja Legoabe
,
Béatrice Josselin
,
Stéphane Bach
,
Sandrine Ruchaud
et al.
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hal-02906292v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
,
Eric Goffin
,
Sebastien Dilly
,
Julien Hanson
,
Lionel Pochet
et al.
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hal-02141338v1
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Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2- a ]pyridines derivatives as protein kinase inhibitors
Marie Lawson
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Jordi Rodrigo
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Blandine Baratte
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Thomas Robert
,
Claire Delehouzé
et al.
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hal-03875851v1
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Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1
Espérance Moine
,
Isabelle Dimier-Poisson
,
Cécile Enguehard-Gueiffier
,
Cédric Logé
,
Mélanie Pénichon
et al.
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hal-02389861v1
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Design and biological evaluation of substituted 5,7-dihydro-6 H -indolo[2,3- c ]quinolin-6-one as novel selective Haspin inhibitors
Sreenivas Avula
,
Xudan Peng
,
Xingfen Lang
,
Micky Tortorella
,
Béatrice Josselin
et al.
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hal-03818922v1
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From simple quinoxalines to potent oxazolo[5,4- f ]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)
Frédéric Lassagne
,
Camille Duguépéroux
,
Carlos Roca
,
Concepcion Perez
,
Ana Martinez
et al.
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hal-03011380v1
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The Anti-Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases
Maciej Masłyk
,
Monika Janeczko
,
Aleksandra Martyna
,
Sławomir Czernik
,
Małgorzata Tokarska-Rodak
et al.
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hal-02046526v1
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Synthesis and Kinase Inhibitory Potencies of Pyrazolo[3,4-g]Isoquinolines
Mathilde Defois
,
Chloé Rémondin
,
Béatrice Josselin
,
Lionel Nauton
,
Vincent Théry
et al.
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hal-03765284v1
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Synthesis and biological evaluation of selected 7H-pyrrolo[2,3-d]pyrimidine derivatives as novel CDK9/CyclinT and Haspin inhibitors
Lianie Pieterse
,
Richard Beteck
,
Blandine Baratte
,
Omobolanle Jesumoroti
,
Thomas Robert
et al.
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hal-03864115v1
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Discovery of simplified benzazole fragments derived from the marine benzosceptrin B as necroptosis inhibitors involving the receptor interacting protein Kinase-1
Mohamed Benchekroun
,
Ludmila Ermolenko
,
Minh Quan Tran
,
Agathe Vagneux
,
Hristo Nedev
et al.
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hal-03004425v2
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Reactivity Under Microwave Irradiation of 2-amino 4H-chromene-3-carbonitrile as tool for the construction of potential bioactive derivatives
Ali Bouattour
,
Mehdi Fakhfakh
,
Houcine Ammar
,
Ludovic Paquin
,
Jean-Pierre Bazureau
et al.
3rd International Electronic Conference on Medicinal Chemistry , Nov 2022, Online, France
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hal-03872422v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
Camille Déliko Dago
,
Christelle Ambeu
,
Wacothon-Karime Coulibaly
,
Yves-Alain Békro
,
Janat Mamyrbékova
et al.
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hal-01187427v1
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
Frédéric Lassagne
,
Timothy Langlais
,
Elsa Caytan
,
Emmanuelle Limanton
,
Ludovic Paquin
et al.
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hal-03867783v1
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Exploration of 7-azaindole-coumaranone hybrids and their analogues as protein kinase inhibitors
Malikotsi Qhobosheane
,
Richard Beteck
,
Blandine Baratte
,
Thomas Robert
,
Sandrine Ruchaud
et al.
Journal articles
hal-03864214v1
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From drug screening to target deconvolution: A target-based drug discovery pipeline using Leishmania casein kinase 1 isoform 2 to identify compounds with anti-leishmanial activity
Emilie Durieu
,
Eric Prina
,
Olivier Leclercq
,
Nassima Oumata
,
Nicolas Gaboriaud-Kolar
et al.
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hal-01299756v1
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Développement de nouveaux inhibiteurs de TgCDPK1 à visée anti-toxoplasmique
Espérance Moine
,
Isabelle Dimier-Poisson
,
Cécile Enguehard-Gueiffier
,
Cedric Logé
,
Mélanie Pénichon
et al.
6. Journées du Consortium antiParasitaire et antiFongique : CaPF-2016 " A la croisée des Mondes !" , Consortium Anti-Parasitaire et Fongique (CaPF). FRA., Mar 2016, Tours, France. 49 p
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hal-02739722v1
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Conception, synthèse et évaluation de nouveaux inhibiteurs de TgCDPK1 à visée anti-toxoplasmique
Espérance Moine
,
Isabelle Dimier-Poisson
,
Cécile Enguehard-Gueiffier
,
Mélanie Pouvreau
,
Nathalie Moiré
et al.
28. Colloque Biotechnocentre , Biotechnocentre. FRA., Oct 2015, Seillac, France
Conference papers
hal-02744066v1
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