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Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure−Activity Relationship Studies
Simon Gonzalez
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Maria Dumitrascuta
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Emilie Eiselt
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Stevany Louis
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Linda Kunze
et al.
Journal articles
hal-03150260v1
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Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases
Astrid Knuhtsen
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Baptiste Legrand
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Olivier van Der Poorten
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Muriel Amblard
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Jean Martinez
et al.
Journal articles
istex
hal-03564349v1
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A bifunctional-biased mu-opioid agonist–neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects
Armand Drieu La Rochelle
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Karel Guillemyn
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Maria Dumitrascuta
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Charlotte Martin
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Valérie Utard
et al.
Journal articles
hal-02368742v1
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Bifunctional Peptide-Based Opioid Agonist–Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic Pain
Karel Guillemyn
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Joanna Starnowska
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Camille Lagard
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Jolanta Dyniewicz
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Ewelina Rojewska
et al.
Journal articles
hal-02993685v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
Jolien de Neve
,
Thomas M. A. Barlow
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Dirk Tourwé
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Frédéric Bihel
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Frédéric Simonin
et al.
Journal articles
hal-03442028v1
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Synthesis of 3-amino-3,4-dihydro-1H-quinolin-2-ones through regioselective palladium-catalyzed intramolecular cyclization
François Hallé
,
Olivier van Der Poorten
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Christelle Doebelin
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Marie Niederst
,
Séverine Schneider
et al.
Journal articles
hal-02290245v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
Jolien de Neve
,
Thomas M A Barlow
,
Dirk Tourwé
,
Frédéric Bihel
,
Frédéric Simonin
et al.
RSC Medicinal Chemistry, 2021
Journal articles
hal-03435229v1
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Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia
Emilie Eiselt
,
Simon Gonzalez
,
Charlotte Martin
,
Magali Chartier
,
Cecilia Betti
et al.
Journal articles
hal-02400886v1
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Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds
Olivier van Der Poorten
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Baptiste Legrand
,
Lubomir Vezenkov
,
Júlia García-Pindado
,
Nadir Bettache
et al.
Journal articles
hal-03564881v1
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Impact of doubling peptide length on in vivo hydrogel stability and sustained drug release
Julie Heremans
,
Lucie Chevillard
,
Morgane Mannes
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Jessica Mangialetto
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Kaat Leroy
et al.
Journal articles
hal-03822784v1
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Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β 2 Adrenergic Receptor Ligands
Charlotte Martin
,
Samuel Moors
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Mia Danielsen
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Cecilia Betti
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Cecilia Fabris
et al.
Journal articles
hal-03025655v1
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χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds
Olivier van Der Poorten
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Robin van den Hauwe
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Emilie Eiselt
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Cecilia Betti
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Karel Guillemyn
et al.
Journal articles
hal-02368778v1
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Harnessing the Anti-Nociceptive Potential of NK2 and NK3 Ligands in the Design of New Multifunctional mu/delta-Opioid Agonist-Neurokinin Antagonist Peptidomimetics
Charlene Gadais
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Justyna Piekielna-Ciesielska
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Jolien de Neve
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Charlotte Martin
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Anna Janecka
et al.
Journal articles
hal-03367748v1
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Insightful Backbone Modifications Preventing Proteolytic Degradation of Neurotensin Analogs Improve NTS1-Induced Protective Hypothermia
Santo Previti
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Mélanie Vivancos
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Emmanuelle Rémond
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Sabrina Beaulieu
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Jean-Michel Longpré
et al.
Journal articles
hal-03022432v1
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Indoloazepinone-Containing Oligomers as Cell-Penetrating (Non)Peptides: Synthesis, Structuration and Internalization
Olivier van Der Poorten
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Baptiste Legrand
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Lubomir Vezenkov
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Jean Martinez
,
Nadir Bettache
et al.
Journal articles
hal-03576982v1
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Identification and Characteristics of Fusion Peptides Derived From Enveloped Viruses
Camille Lozada
,
Thomas M A Barlow
,
Simon Gonzalez
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Nadège Lubin-Germain
,
Steven Ballet
et al.
Journal articles
hal-03714204v1
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