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authFullName_s : Steven Ballet
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Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure−Activity Relationship Studies

Simon Gonzalez , Maria Dumitrascuta , Emilie Eiselt , Stevany Louis , Linda Kunze et al.
Journal of Medicinal Chemistry, 2020, 63 (21), pp.12929-12941. ⟨10.1021/acs.jmedchem.0c01376⟩
Journal articles hal-03150260v1

Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases

Astrid Knuhtsen , Baptiste Legrand , Olivier van Der Poorten , Muriel Amblard , Jean Martinez et al.
Chemistry - A European Journal, 2016, 22 (39), pp.14022-14028. ⟨10.1002/chem.201602518⟩
Journal articles istex hal-03564349v1

A bifunctional-biased mu-opioid agonist–neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects

Armand Drieu La Rochelle , Karel Guillemyn , Maria Dumitrascuta , Charlotte Martin , Valérie Utard et al.
PAIN, 2018, 159 (9), pp.1705-1718. ⟨10.1097/j.pain.0000000000001262⟩
Journal articles hal-02368742v1
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Bifunctional Peptide-Based Opioid Agonist–Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic Pain

Karel Guillemyn , Joanna Starnowska , Camille Lagard , Jolanta Dyniewicz , Ewelina Rojewska et al.
Journal of Medicinal Chemistry, 2016, 59 (8), pp.3777-3792. ⟨10.1021/acs.jmedchem.5b01976⟩
Journal articles hal-02993685v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors

Jolien de Neve , Thomas M. A. Barlow , Dirk Tourwé , Frédéric Bihel , Frédéric Simonin et al.
RSC Medicinal Chemistry, 2021, 12 (6), pp.828-870. ⟨10.1039/D1MD00041A⟩
Journal articles hal-03442028v1

Synthesis of 3-amino-3,4-dihydro-1H-quinolin-2-ones through regioselective palladium-catalyzed intramolecular cyclization

François Hallé , Olivier van Der Poorten , Christelle Doebelin , Marie Niederst , Séverine Schneider et al.
Tetrahedron Letters, 2016, 57 (14), pp.1547-1550. ⟨10.1016/j.tetlet.2016.02.094⟩
Journal articles hal-02290245v1
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors

Jolien de Neve , Thomas M A Barlow , Dirk Tourwé , Frédéric Bihel , Frédéric Simonin et al.
RSC Medicinal Chemistry, 2021
Journal articles hal-03435229v1

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

Emilie Eiselt , Simon Gonzalez , Charlotte Martin , Magali Chartier , Cecilia Betti et al.
ACS Chemical Neuroscience, 2019, 10 (11), pp.4535-4544. ⟨10.1021/acschemneuro.9b00390⟩
Journal articles hal-02400886v1

Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain-Barrier-Permeating Compounds

Olivier van Der Poorten , Baptiste Legrand , Lubomir Vezenkov , Júlia García-Pindado , Nadir Bettache et al.
ChemBioChem, 2018, 19 (7), pp.696-705. ⟨10.1002/cbic.201700678⟩
Journal articles hal-03564881v1

Impact of doubling peptide length on in vivo hydrogel stability and sustained drug release

Julie Heremans , Lucie Chevillard , Morgane Mannes , Jessica Mangialetto , Kaat Leroy et al.
Journal of Controlled Release, 2022, 350, pp.514-524. ⟨10.1016/j.jconrel.2022.08.027⟩
Journal articles hal-03822784v1

Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β 2 Adrenergic Receptor Ligands

Charlotte Martin , Samuel Moors , Mia Danielsen , Cecilia Betti , Cecilia Fabris et al.
Chemistry - A European Journal, 2017, 23 (40), pp.9632-9640. ⟨10.1002/chem.201701321⟩
Journal articles hal-03025655v1

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds

Olivier van Der Poorten , Robin van den Hauwe , Emilie Eiselt , Cecilia Betti , Karel Guillemyn et al.
ACS Medicinal Chemistry Letters, 2017, 8 (11), pp.1177-1182. ⟨10.1021/acsmedchemlett.7b00347⟩
Journal articles hal-02368778v1
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Harnessing the Anti-Nociceptive Potential of NK2 and NK3 Ligands in the Design of New Multifunctional mu/delta-Opioid Agonist-Neurokinin Antagonist Peptidomimetics

Charlene Gadais , Justyna Piekielna-Ciesielska , Jolien de Neve , Charlotte Martin , Anna Janecka et al.
Molecules, 2021, 26 (17), pp.5406. ⟨10.3390/molecules26175406⟩
Journal articles hal-03367748v1
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Insightful Backbone Modifications Preventing Proteolytic Degradation of Neurotensin Analogs Improve NTS1-Induced Protective Hypothermia

Santo Previti , Mélanie Vivancos , Emmanuelle Rémond , Sabrina Beaulieu , Jean-Michel Longpré et al.
Frontiers in Chemistry, 2020, ⟨10.3389/fchem.2020.00406⟩
Journal articles hal-03022432v1

Indoloazepinone-Containing Oligomers as Cell-Penetrating (Non)Peptides: Synthesis, Structuration and Internalization

Olivier van Der Poorten , Baptiste Legrand , Lubomir Vezenkov , Jean Martinez , Nadir Bettache et al.
Journal of Peptide Science, 2018, 22 (S2), pp.S117. ⟨10.1002/psc.2950⟩
Journal articles hal-03576982v1
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Identification and Characteristics of Fusion Peptides Derived From Enveloped Viruses

Camille Lozada , Thomas M A Barlow , Simon Gonzalez , Nadège Lubin-Germain , Steven Ballet et al.
Frontiers in Chemistry, 2022, 12, pp.689006. ⟨10.3389/fchem.2021.689006⟩
Journal articles hal-03714204v1