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authFullName_s : Vittorio Canale

The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3

Paweł Zajdel , Nicolas Masurier , Vittorio Canale , Pascal Verdie , Muriel Amblard et al.
Tetrahedron Letters, 2013, 54 (8), pp.998-1002. ⟨10.1016/j.tetlet.2012.12.036⟩
Journal articles hal-03563368v1
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mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatment

Pierre-Yves Martin , Stéphane Doly , Al Mahdy Hamieh , Eric Chapuy , Vittorio Canale et al.
Progress in Neurobiology, 2020, 193, pp.101846. ⟨10.1016/j.pneurobio.2020.101846⟩
Journal articles hal-02906397v1
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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity

Vittorio Canale , Wojciech Trybała , Séverine Chaumont-Dubel , Paulina Koczurkiewicz-Adamczyk , Grzegorz Satała et al.
Biomolecules, 2023, 13 (1), pp.12. ⟨10.3390/biom13010012⟩
Journal articles hal-03933561v1

Novel non-sulfonamide 5-HT 6 receptor partial inverse agonist in a group of imidazo[4,5- b ]pyridines with cognition enhancing properties

David Vanda , Miroslav Soural , Vittorio Canale , Séverine Chaumont-Dubel , Grzegorz Satała et al.
European Journal of Medicinal Chemistry, 2018, 144, pp.716-729. ⟨10.1016/j.ejmech.2017.12.053⟩
Journal articles hal-02366387v1
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Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties

Vittorio Canale , Magdalena Kotańska , Anna Dziubina , Matylda Stefaniak , Agata Siwek et al.
Molecules, 2021, 26 (13), pp.3828. ⟨10.3390/molecules26133828⟩
Journal articles hal-03269422v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties

Vittorio Canale , Katarzyna Grychowska , Rafał Kurczab , Mateusz Ryng , Abdul Raheem Keeri et al.
European Journal of Medicinal Chemistry, 2020, 208, pp.112765. ⟨10.1016/j.ejmech.2020.112765⟩
Journal articles hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity

Marcin Drop , Vittorio Canale , Séverine Chaumont-Dubel , Rafał Kurczab , Grzegorz Satała et al.
ACS Chemical Neuroscience, 2021, 12 (7), pp.1228-1240. ⟨10.1021/acschemneuro.1c00061⟩
Journal articles hal-03192567v1
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Sustainable Synthesis of a Potent and Selective 5-HT7 Receptor Antagonist Using a Mechanochemical Approach

Vittorio Canale , Valeria Frisi , Xavier Bantreil , Frédéric Lamaty , Paweł Zajdel et al.
Journal of Organic Chemistry, 2020, 85 (16), pp.10958-10965. ⟨10.1021/acs.joc.0c01044⟩
Journal articles hal-02925108v1

Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands

Vittorio Canale , Paweł Guzik , Rafał Kurczab , Pascal Verdie , Grzegorz Satała et al.
European Journal of Medicinal Chemistry, 2014, 78, pp.10-22. ⟨10.1016/j.ejmech.2014.03.005⟩
Journal articles hal-03563396v1
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Neuropathic pain-alleviating activity of novel 5-HT6 receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide

Marcin Drop , Florian Jacquot , Vittorio Canale , Séverine Chaumont-Dubel , Maria Walczak et al.
Bioorganic Chemistry, 2021, 115, pp.105218. ⟨10.1016/j.bioorg.2021.105218⟩
Journal articles hal-03324439v1
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The Constitutive Activity of Spinal 5-HT6 Receptors Contributes to Diabetic Neuropathic Pain in Rats

Nazarine Mokhtar , Marcin Drop , Florian Jacquot , Sylvain Lamoine , Eric Chapuy et al.
Biomolecules, 2023, 13 (2), pp.364. ⟨10.3390/biom13020364⟩
Journal articles hal-03996855v1