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The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3
Paweł Zajdel
,
Nicolas Masurier
,
Vittorio Canale
,
Pascal Verdie
,
Muriel Amblard
et al.
Journal articles
hal-03563368v1
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mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatment
Pierre-Yves Martin
,
Stéphane Doly
,
Al Mahdy Hamieh
,
Eric Chapuy
,
Vittorio Canale
et al.
Journal articles
hal-02906397v1
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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity
Vittorio Canale
,
Wojciech Trybała
,
Séverine Chaumont-Dubel
,
Paulina Koczurkiewicz-Adamczyk
,
Grzegorz Satała
et al.
Journal articles
hal-03933561v1
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Novel non-sulfonamide 5-HT 6 receptor partial inverse agonist in a group of imidazo[4,5- b ]pyridines with cognition enhancing properties
David Vanda
,
Miroslav Soural
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Grzegorz Satała
et al.
Journal articles
hal-02366387v1
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Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties
Vittorio Canale
,
Magdalena Kotańska
,
Anna Dziubina
,
Matylda Stefaniak
,
Agata Siwek
et al.
Journal articles
hal-03269422v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
Vittorio Canale
,
Katarzyna Grychowska
,
Rafał Kurczab
,
Mateusz Ryng
,
Abdul Raheem Keeri
et al.
Journal articles
hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity
Marcin Drop
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Grzegorz Satała
et al.
Journal articles
hal-03192567v1
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Sustainable Synthesis of a Potent and Selective 5-HT7 Receptor Antagonist Using a Mechanochemical Approach
Vittorio Canale
,
Valeria Frisi
,
Xavier Bantreil
,
Frédéric Lamaty
,
Paweł Zajdel
et al.
Journal articles
hal-02925108v1
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Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT7 and 5-HT1A receptor ligands
Vittorio Canale
,
Paweł Guzik
,
Rafał Kurczab
,
Pascal Verdie
,
Grzegorz Satała
et al.
Journal articles
hal-03563396v1
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Neuropathic pain-alleviating activity of novel 5-HT6 receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide
Marcin Drop
,
Florian Jacquot
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Maria Walczak
et al.
Journal articles
hal-03324439v1
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The Constitutive Activity of Spinal 5-HT6 Receptors Contributes to Diabetic Neuropathic Pain in Rats
Nazarine Mokhtar
,
Marcin Drop
,
Florian Jacquot
,
Sylvain Lamoine
,
Eric Chapuy
et al.
Journal articles
hal-03996855v1
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