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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity

Vittorio Canale , Wojciech Trybała , Séverine Chaumont-Dubel , Paulina Koczurkiewicz-Adamczyk , Grzegorz Satała et al.
Biomolecules, 2023, 13 (1), pp.12. ⟨10.3390/biom13010012⟩
Journal articles hal-03933561v1
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Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties

Vittorio Canale , Magdalena Kotańska , Anna Dziubina , Matylda Stefaniak , Agata Siwek et al.
Molecules, 2021, 26 (13), pp.3828. ⟨10.3390/molecules26133828⟩
Journal articles hal-03269422v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties

Vittorio Canale , Katarzyna Grychowska , Rafał Kurczab , Mateusz Ryng , Abdul Raheem Keeri et al.
European Journal of Medicinal Chemistry, 2020, 208, pp.112765. ⟨10.1016/j.ejmech.2020.112765⟩
Journal articles hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity

Marcin Drop , Vittorio Canale , Séverine Chaumont-Dubel , Rafał Kurczab , Grzegorz Satała et al.
ACS Chemical Neuroscience, 2021, 12 (7), pp.1228-1240. ⟨10.1021/acschemneuro.1c00061⟩
Journal articles hal-03192567v1
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Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-pyrrolo[3,2-c]quinoline Series

Katarzyna Grychowska , Wojciech Pietruś , Ludmiła Kulawik , Ophélie Bento , Grzegorz Satała et al.
Molecules, 2023, 28, pp.1096. ⟨10.3390/molecules28031096⟩
Journal articles hal-03956220v1
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Blockade of Serotonin 5-HT6 Receptor Constitutive Activity Alleviates Cognitive Deficits in a Preclinical Model of Neurofibromatosis Type 1

Emilie Doucet , Katarzyna Grychowska , Pawel Zajdel , Joël Bockaert , Philippe Marin et al.
International Journal of Molecular Sciences, 2021, 22 (18), pp.10178. ⟨10.3390/ijms221810178⟩
Journal articles hal-03801130v1
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The Constitutive Activity of Spinal 5-HT6 Receptors Contributes to Diabetic Neuropathic Pain in Rats

Nazarine Mokhtar , Marcin Drop , Florian Jacquot , Sylvain Lamoine , Eric Chapuy et al.
Biomolecules, 2023, 13 (2), pp.364. ⟨10.3390/biom13020364⟩
Journal articles hal-03996855v1
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Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity

Katarzyna Grychowska , Séverine Chaumont-Dubel , Rafał Kurczab , Paulina Koczurkiewicz , Caroline Deville et al.
ACS Chemical Neuroscience, 2019, 10 (7), pp.3183-3196. ⟨10.1021/acschemneuro.8b00618⟩
Journal articles hal-02364291v1