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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity
Vittorio Canale
,
Wojciech Trybała
,
Séverine Chaumont-Dubel
,
Paulina Koczurkiewicz-Adamczyk
,
Grzegorz Satała
et al.
Journal articles
hal-03933561v1
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Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties
Vittorio Canale
,
Magdalena Kotańska
,
Anna Dziubina
,
Matylda Stefaniak
,
Agata Siwek
et al.
Journal articles
hal-03269422v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
Vittorio Canale
,
Katarzyna Grychowska
,
Rafał Kurczab
,
Mateusz Ryng
,
Abdul Raheem Keeri
et al.
Journal articles
hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity
Marcin Drop
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Grzegorz Satała
et al.
Journal articles
hal-03192567v1
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Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-pyrrolo[3,2-c]quinoline Series
Katarzyna Grychowska
,
Wojciech Pietruś
,
Ludmiła Kulawik
,
Ophélie Bento
,
Grzegorz Satała
et al.
Journal articles
hal-03956220v1
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Blockade of Serotonin 5-HT6 Receptor Constitutive Activity Alleviates Cognitive Deficits in a Preclinical Model of Neurofibromatosis Type 1
Emilie Doucet
,
Katarzyna Grychowska
,
Pawel Zajdel
,
Joël Bockaert
,
Philippe Marin
et al.
Journal articles
hal-03801130v1
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The Constitutive Activity of Spinal 5-HT6 Receptors Contributes to Diabetic Neuropathic Pain in Rats
Nazarine Mokhtar
,
Marcin Drop
,
Florian Jacquot
,
Sylvain Lamoine
,
Eric Chapuy
et al.
Journal articles
hal-03996855v1
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Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity
Katarzyna Grychowska
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Paulina Koczurkiewicz
,
Caroline Deville
et al.
Journal articles
hal-02364291v1
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