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Solid-Supported Synthesis and 5-HT 7 /5-HT 1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H )-one

Katarzyna Grychowska , Nicolas Masurier , Pascal Verdié , Grzegorz Satała , Andrzej Bojarski et al.
Chemical Biology and Drug Design, 2015, 86 (4), pp.697-703. ⟨10.1111/cbdd.12539⟩
Journal articles istex hal-03564059v1
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Application of the ring-closing metathesis to the formation of 2-aryl-1 H -pyrrole-3-carboxylates as building blocks for biologically active compounds

Katarzyna Grychowska , B. Kubica , Marcin Drop , Evelina Colacino , Xavier Bantreil et al.
Tetrahedron, 2016, 72 (47), pp.7462-7469. ⟨10.1016/j.tet.2016.09.059⟩
Journal articles hal-02385423v1
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Early 5‐ HT 6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse

Coralie Berthoux , Al Mahdy Hamieh , Angelina Rogliardo , Emilie Doucet , Camille Coudert et al.
EMBO Molecular Medicine, 2020, 12 (5), pp.e10605. ⟨10.15252/emmm.201910605⟩
Journal articles hal-02863763v1
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Continuous flow ring-closing metathesis, an environmentally-friendly route to 2,5-dihydro-1H-pyrrole-3-carboxylates

Marcin Drop , Xavier Bantreil , Katarzyna Grychowska , Gilbert Umuhire Mahoro , Evelina Colacino et al.
Green Chemistry, 2017, 19 (7), pp.1647-1652. ⟨10.1039/c7gc00235a⟩
Journal articles hal-02385309v1
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Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT 3 and 5-HT 6 Receptor Antagonist with Antipsychotic and Procognitive Properties

Paweł Zajdel , Katarzyna Grychowska , Szczepan Mogilski , Rafał Kurczab , Grzegorz Satała et al.
Journal of Medicinal Chemistry, 2021, 64 (18), pp.13279-13298. ⟨10.1021/acs.jmedchem.1c00224⟩
Journal articles hal-03357806v1
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Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines

Katarzyna Grychowska , Agnieszka Olejarz-Maciej , Klaudia Blicharz , Wojciech Pietruś , Tadeusz Karcz et al.
European Journal of Medicinal Chemistry, 2022, 236, pp.114329. ⟨10.1016/j.ejmech.2022.114329⟩
Journal articles hal-03648220v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties

Vittorio Canale , Katarzyna Grychowska , Rafał Kurczab , Mateusz Ryng , Abdul Raheem Keeri et al.
European Journal of Medicinal Chemistry, 2020, 208, pp.112765. ⟨10.1016/j.ejmech.2020.112765⟩
Journal articles hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity

Marcin Drop , Vittorio Canale , Séverine Chaumont-Dubel , Rafał Kurczab , Grzegorz Satała et al.
ACS Chemical Neuroscience, 2021, 12 (7), pp.1228-1240. ⟨10.1021/acschemneuro.1c00061⟩
Journal articles hal-03192567v1
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Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease

Katarzyna Grychowska , Grzegorz Satala , Tomasz Kos , Anna Partyka , Evelina Colacino et al.
ACS Chemical Neuroscience, 2016, 7 (7), pp.972--83. ⟨10.1021/acschemneuro.6b00090⟩
Journal articles hal-01941175v1
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Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity

Katarzyna Grychowska , Séverine Chaumont-Dubel , Rafał Kurczab , Paulina Koczurkiewicz , Caroline Deville et al.
ACS Chemical Neuroscience, 2019, 10 (7), pp.3183-3196. ⟨10.1021/acschemneuro.8b00618⟩
Journal articles hal-02364291v1