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Solid-Supported Synthesis and 5-HT 7 /5-HT 1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H )-one
Katarzyna Grychowska
,
Nicolas Masurier
,
Pascal Verdié
,
Grzegorz Satała
,
Andrzej Bojarski
et al.
Journal articles
istex
hal-03564059v1
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Application of the ring-closing metathesis to the formation of 2-aryl-1 H -pyrrole-3-carboxylates as building blocks for biologically active compounds
Katarzyna Grychowska
,
B. Kubica
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Marcin Drop
,
Evelina Colacino
,
Xavier Bantreil
et al.
Journal articles
hal-02385423v1
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Early 5‐ HT 6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse
Coralie Berthoux
,
Al Mahdy Hamieh
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Angelina Rogliardo
,
Emilie Doucet
,
Camille Coudert
et al.
Journal articles
hal-02863763v1
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Continuous flow ring-closing metathesis, an environmentally-friendly route to 2,5-dihydro-1H-pyrrole-3-carboxylates
Marcin Drop
,
Xavier Bantreil
,
Katarzyna Grychowska
,
Gilbert Umuhire Mahoro
,
Evelina Colacino
et al.
Journal articles
hal-02385309v1
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Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT 3 and 5-HT 6 Receptor Antagonist with Antipsychotic and Procognitive Properties
Paweł Zajdel
,
Katarzyna Grychowska
,
Szczepan Mogilski
,
Rafał Kurczab
,
Grzegorz Satała
et al.
Journal articles
hal-03357806v1
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Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c]quinolines
Katarzyna Grychowska
,
Agnieszka Olejarz-Maciej
,
Klaudia Blicharz
,
Wojciech Pietruś
,
Tadeusz Karcz
et al.
Journal articles
hal-03648220v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
Vittorio Canale
,
Katarzyna Grychowska
,
Rafał Kurczab
,
Mateusz Ryng
,
Abdul Raheem Keeri
et al.
Journal articles
hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity
Marcin Drop
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Grzegorz Satała
et al.
Journal articles
hal-03192567v1
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Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease
Katarzyna Grychowska
,
Grzegorz Satala
,
Tomasz Kos
,
Anna Partyka
,
Evelina Colacino
et al.
Journal articles
hal-01941175v1
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Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity
Katarzyna Grychowska
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Paulina Koczurkiewicz
,
Caroline Deville
et al.
Journal articles
hal-02364291v1
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