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NMR tool for the characterization of protein-fragment complexes
Olivier Cala
,
Clémentine Aguirre
,
Tim Ten Brink
,
Isabelle Krimm
GERM XXV - Conférence du Groupe Français d'Etude de Résonance Magnétique, Jun 2014, Biarritz, France
Conference papers
hal-01018840v1
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INPHARMA-based identification of ligand binding site in fragment-based drug design
Isabelle Krimm
Journal articles
hal-00819132v1
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NMR-Based Characterization of Protein-Fragment Complexes
Isabelle Krimm
Discovery Chemistry Congress, Mar 2013, Munich, Germany
Conference papers
hal-00819152v1
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Tackling the Interaction of the Multidomain Protein STAM2 with Ubiquitin and Diubiquitin Chains by NMR. Cooperativity or not, that is the Question !
Florence Guillière
,
Jean-Marc Lancelin
,
Isabelle Krimm
,
Olivier Walker
,
Anja Lange
et al.
XXVth International Conference on Magnetic Resonance in Biological Systems (ICMRBS), Aug 2012, Lyon, France
Conference papers
hal-00958296v1
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Performance of Protein–Ligand Docking with Simulated Chemical Shift Perturbations
Tim Ten Brink
,
Clémentine Aguirre
,
Thomas E. Exner
,
Isabelle Krimm
Journal articles
hal-01087991v1
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Fragment Linking Strategies for Structure-Based Drug Design
Alexandre Bancet
,
Claire Raingeval
,
Thierry Lomberget
,
Marc Le Borgne
,
Jean-François Guichou
et al.
Journal articles
hal-03045139v1
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NMR for Fragment-Based Drug Design
Olivier Cala
,
Isabelle Krimm
27th International Conference on Magnetic Resonance in Biological Systems - ICMRBS2016, Aug 2016, Kyoto, Japan
Conference poster
hal-01397732v1
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Miniaturized weak affinity chromatography for ligand identification of nanodiscs-embedded G-protein coupled receptors
Lucile Lecas
,
Lucie Hartmann
,
Lydia Caro
,
Sarah Mohamed-Bouteben
,
Claire Raingeval
et al.
Journal articles
hal-03045118v1
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Comparing Binding Modes of Analogous Fragments Using NMR in Fragment-Based Drug Design: Application to PRDX5
Clémentine Aguirre
,
Tim Ten Brink
,
Jean François Guichou
,
Olivier Cala
,
Isabelle Krimm
et al.
Journal articles
hal-01067905v1
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Comparaison du mode de liaison de fragments analogues par RMN quantitative dans le contexte du Drug Design
Clémentine Aguirre
,
Tim Ten Brink
,
Olivier Cala
,
Isabelle Krimm
15ème Journée RMN Rhône Alpes, Jun 2014, Grenoble, France
Conference papers
hal-01018842v1
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NMR applications in FBDD regarding fragment binding mode and framgent-induced protein conformational change
Isabelle Krimm
Zing Conference - Fragment-Based Drug Discovery, Jul 2014, Punta Cana, Dominican Republic
Conference papers
hal-00955950v1
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Les molécules fragments : un outil puissant en chimie biologique
Isabelle Krimm
14èmes REncontres en Chimie Organique Biologique (RECOB'14), Mar 2012, Aussois, France
Conference papers
hal-00819219v1
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Protein–ligand structure guided by backbone and side-chain proton chemical shift perturbations
Clémentine Aguirre
,
Olivier Cala
,
Tim Ten Brink
,
Jean François Guichou
,
Isabelle Krimm
et al.
Journal articles
hal-01088012v1
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Fragment-based screening: a promising avenue for drug design
Isabelle Krimm
Journal articles
hal-01187367v1
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HalX: an open-source LIMS (Laboratory Information Management System) for small- to large-scale laboratories.
Jaime Prilusky
,
Eric Oeuillet
,
Nathalie Ulryck
,
Anne Pajon
,
Julie Bernauer
et al.
Journal articles
istex
inria-00431702v1
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Etude de complexes protéine-ligand par RMN quantitative dans le contexte du Drug Design
Clémentine Aguirre
,
Florence Guillière
,
Dany Davesne
,
Isabelle Krimm
Journée de Printemps de la Société Chimique de France, Jun 2012, Lyon, France
Conference papers
hal-00819230v1
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A Deep Dive into VDAC1 Conformational Diversity Using All-Atom Simulations Provides New Insights into the Structural Origin of the Closed States
Jordane Preto
,
Hubert Gorny
,
Isabelle Krimm
Journal articles
hal-03856956v1
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Biophysical Dissection of Isolated GPCRs: The Adenosine A2A Receptor under the Bistouries
Jean-Louis Banères
,
Thomas Botzanowski
,
Jean A Boutin
,
Barbara Calamini
,
Jérôme Castel
et al.
Journal articles
hal-04003751v1
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Probing ligand binding mode by NMR in Fragment-Based Drug design
Clémentine Aguirre
,
Florence Guillière
,
Dany Davesne
,
Isabelle Krimm
XXVth International Conference on Magnetic Resonance in Biological Systems (ICMRBS), Aug 2012, Lyon, France
Conference papers
hal-00819174v1
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Probing hot spots on protein-protein interfaces using fragment-based drug design
Sarah Barelier
,
Isabelle Krimm
EMBO Workshop "Advances in Protein-Protein - Interaction Analysis & Modulation", Jun 2012, Roscoff, France
Conference papers
hal-00819202v1
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Etude de complexes protéine-ligand par RMN quantitative dans le contexte du Drug Design
Clémentine Aguirre
,
Isabelle Krimm
GTBio 2012, Apr 2012, Montpellier, France
Conference papers
hal-00819210v1
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Analyse des complexes protéine-ligand par RMN dans le cadre de la conception de médicaments
Clémentine Aguirre
,
Tim Ten Brink
,
Isabelle Krimm
Journée Rhône-Alpes des Biomolécules (JRAB 2013), Jun 2013, Lyon, France
Conference papers
hal-00873777v1
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Applications of NMR for fragment-based drug design
Isabelle Krimm
,
Olivier Cala
Journée scientifique de la Fédération de Recherche FR2708 (COA UMR 7311 et CBM UPR4301), Jun 2014, Orléans, France
Conference papers
hal-01067919v1
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1D NMR WaterLOGSY as an efficient method for fragment-based lead discovery
Claire Raingeval
,
Olivier Cala
,
Béatrice Brion
,
Marc Le Borgne
,
Roderick Eliot Hubbard
et al.
Journal articles
hal-02188259v1
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Evolution et nouvelles tendances dans les sciences analytiques pour le domaine pharmaceutique
Isabelle Krimm
Congrès Africain et Francophone sur les Sciences Analytiques et Applications (CAFSAA) , Nov 2017, Hammamet, Tunisie
Conference papers
hal-01864864v1
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NMR structures of thioredoxin m from the green alga Chlamydomonas reinhardtii
Jean‐marc Lancelin
,
Laure Guilhaudis
,
Isabelle Krimm
,
Martin Blackledge
,
Dominique Marion
et al.
Journal articles
hal-02352003v1
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A Combination of Spin Diffusion Methods for the Determination of Protein-Ligand Complex Structural Ensembles
Jens Pilger
,
Adam Mazur
,
Peter Monecke
,
Herman Schreuder
,
Bettina Elshorst
et al.
Journal articles
istex
hal-01165216v1
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NMR approaches in fragment-based drug design
Isabelle Krimm
ChemBioInteract "Conference on Drug Discovery & Drug Design: ChemBio Interactions", Oct 2013, Lyon, France
Conference papers
hal-00955939v1
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BcL-xL Conformational Changes upon Fragment Binding Revealed by NMR
Clémentine Aguirre
,
Tim Ten Brink
,
Olivier Walker
,
Florence Guillière
,
D. Davesne
et al.
Journal articles
in2p3-00839023v1
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The Dynamics of Copper Uptake in Human Cu,Zn-Superoxide Dismutase: a Solid-State NMR Study
Claire Raingeval
,
Olivier Cala
,
Béatrice Brion
,
Isabelle Krimm
XXIXème congrès du GERM, Groupement d'études de résonance magnétique, May 2017, Aussois, France
Conference papers
hal-01865374v1
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