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authIdHal_s : philippe-robert-marin
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Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT 3 and 5-HT 6 Receptor Antagonist with Antipsychotic and Procognitive Properties

Paweł Zajdel , Katarzyna Grychowska , Szczepan Mogilski , Rafał Kurczab , Grzegorz Satała et al.
Journal of Medicinal Chemistry, 2021, 64 (18), pp.13279-13298. ⟨10.1021/acs.jmedchem.1c00224⟩
Journal articles hal-03357806v1

Cdk5 induces constitutive activation of 5-HT6 receptors to promote neurite growth

Fanny Duhr , Paul Déléris , F. Raynaud , Martial Séveno , Séverine Morisset-Lopez et al.
Nature Chemical Biology, 2014, 10 (7), pp.590-597. ⟨10.1038/nchembio.1547⟩
Journal articles hal-01178901v1

5 HT4 agonists: novel promising agents for AD prevention.

Patrizia Giannoni , Florence Gaven , Kévin Baranger , Santiago Rivera , Philippe Marin et al.
AD/PD 2013, Mar 2013, Florence, Italy
Conference poster hal-02918547v1
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The serotonin 6 receptor controls neuronal migration during corticogenesis via a ligand-independent Cdk5-dependent mechanism

M. Jacobshagen , M. Niquille , Séverine Chaumont-Dubel , Philippe Marin , A. Dayer et al.
Development (Cambridge, England), 2014, 141 (17), pp.3370--7. ⟨10.1242/dev.108043⟩
Journal articles hal-01950135v1
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Presynaptic serotonin 2A receptors modulate thalamocortical plasticity and associative learning

Alexander Barre , Coralie Berthoux , Dimitri de Bundel , Emmanuel Valjent , Joël Bockaert et al.
Proceedings of the National Academy of Sciences of the United States of America, 2016, 113 (10), pp.E1382--91. ⟨10.1073/pnas.1525586113⟩
Journal articles hal-01942458v1
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The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release

Jérémie Neasta , Charlène Valmalle , Anne‐claire Coyne , Eric Carnazzi , Gilles Subra et al.
British Journal of Pharmacology, 2016, 173 (8), pp.1314--28. ⟨10.1111/bph.13424⟩
Journal articles hal-01942451v1

5 HT4 agonists: novel promising agents for AD prevention.

Patrizia Giannoni , Florence Gaven , Kévin Baranger , Santiago Rivera , Philippe Marin et al.
Congrès des Neurosciences Francaises, May 2013, Lyon, France
Conference poster hal-02918543v1
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mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatment

Pierre-Yves Martin , Stéphane Doly , Al Mahdy Hamieh , Eric Chapuy , Vittorio Canale et al.
Progress in Neurobiology, 2020, 193, pp.101846. ⟨10.1016/j.pneurobio.2020.101846⟩
Journal articles hal-02906397v1
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Early 5‐ HT 6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse

Coralie Berthoux , Al Mahdy Hamieh , Angelina Rogliardo , Emilie Doucet , Camille Coudert et al.
EMBO Molecular Medicine, 2020, 12 (5), pp.e10605. ⟨10.15252/emmm.201910605⟩
Journal articles hal-02863763v1
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Dynamic interactions of the 5-HT 6 receptor with protein partners control dendritic tree morphogenesis

Camille Pujol , Vincent Dupuy , Martial Séveno , Léonie Runtz , Joël Bockaert et al.
Science Signaling, 2020, 13 (618), pp.eaax9520. ⟨10.1126/scisignal.aax9520⟩
Journal articles hal-02485360v1
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Shank3-Rich2 Interaction Regulates AMPA Receptor Recycling and Synaptic Long-Term Potentiation

F. Raynaud , A. Janossy , J. Dahl , F. Bertaso , J. Perroy et al.
Journal of Neuroscience, 2013, 33 (23), pp.9699-9715. ⟨10.1523/JNEUROSCI.2725-12.2013⟩
Journal articles hal-02309091v1
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Novel and atypical pathways for serotonin signaling

Joël Bockaert , Carine Becamel , Séverine Chaumont-Dubel , Sylvie Claeysen , Franck Vandermoere et al.
Faculty Reviews, 2021, 10, pp.52. ⟨10.12703/r/10-52⟩
Journal articles hal-03256253v1
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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity

Vittorio Canale , Wojciech Trybała , Séverine Chaumont-Dubel , Paulina Koczurkiewicz-Adamczyk , Grzegorz Satała et al.
Biomolecules, 2023, 13 (1), pp.12. ⟨10.3390/biom13010012⟩
Journal articles hal-03933561v1
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Spatiotemporal dynamics of 5-HT6 receptor ciliary localization during mouse brain development

Vincent Dupuy , Matthieu Prieur , Anne Pizzoccaro , Clara Margarido , Emmanuel Valjent et al.
Neurobiology of Disease, 2022, 176, pp.105949. ⟨10.1016/j.nbd.2022.105949⟩
Journal articles hal-03900095v1

Co-assembly of two GluR6 kainate receptor splice variants within a functional protein complex

F. Coussen , D. Perrais , F. Jaskolski , S. Sachidhanandam , E. Normand et al.
Neuron, 2005, 47, pp.555-566. ⟨10.1016/j.neuron.2005.06.033⟩
Journal articles hal-00016946v1

p.N680S single nucleotide polymorphism of the FSHR affects FSH-induced β-arrestin recruitment, β-arrestin-dependent translocation of PKA catalytic subunit to the nucleus and CRE-driven transcription

Flavie Landomiel , Thibaud Tranchant , Guillaume Durand , Alfredo Ulloa Aguirre , Pascale Crépieux et al.
International Conference on Gonadotropins & Receptors, Sep 2014, Tours, France. , 2014, ICGRIII International Conference on Gonadotropins & Receptors
Conference poster hal-02739343v1

Novel non-sulfonamide 5-HT 6 receptor partial inverse agonist in a group of imidazo[4,5- b ]pyridines with cognition enhancing properties

David Vanda , Miroslav Soural , Vittorio Canale , Séverine Chaumont-Dubel , Grzegorz Satała et al.
European Journal of Medicinal Chemistry, 2018, 144, pp.716-729. ⟨10.1016/j.ejmech.2017.12.053⟩
Journal articles hal-02366387v1
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Quantitative Phosphoproteomics Unravels Biased Phosphorylation of Serotonin 2A Receptor at Ser 280 by Hallucinogenic versus Nonhallucinogenic Agonists

Samah Karaki , Carine Becamel , Samy Murat , Clotilde Mannoury La Cour , Mark Millan et al.
Molecular and Cellular Proteomics, 2014, 13 (5), pp.1273-1285. ⟨10.1074/mcp.M113.036558⟩
Journal articles hal-02366017v1

Physical and functional interactions between the serotonin transporter and the neutral amino acid transporter ASCT2

Pascal Seyer , Franck Vandermoere , Elisabeth Cassier , Joël Bockaert , Philippe Marin et al.
Biochemical Journal, 2016, 473 (13), pp.1953--65. ⟨10.1042/BCJ20160315⟩
Journal articles hal-01941172v1

New insights in molecular aspects of Alzheimer’s disease. Conférencière invitée.

Patrizia Giannoni , Florence Gaven , Kévin Baranger , Santiago Rivera , Philippe Marin et al.
Sindem, Mar 2013, Perugia, Italy
Conference papers hal-02918588v1
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Effects of a psychedelic 5-HT2A receptor agonist on anxiety-related behavior and fear processing in mice

Błażej Pędzich , Sarah Rubens , Mehdi Sekssaoui , Anouk Pierre , Andries van Schuerbeek et al.
Neuropsychopharmacology, 2022, 47 (7), pp.1304-1314. ⟨10.1038/s41386-022-01324-2⟩
Journal articles hal-03653250v1
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Differentiated glioma cell-derived fibromodulin activates integrin-dependent Notch signaling in endothelial cells to promote tumor angiogenesis and growth

Shreoshi Sengupta , Mainak Mondal , Kaval Reddy Prasasvi , Arani Mukherjee , Prerna Magod et al.
eLife, 2022, 11, pp.e78972. ⟨10.7554/eLife.78972⟩
Journal articles hal-03755078v1
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Amelioration of Tau pathology and memory deficits by targeting 5-HT7 receptor

Josephine Labus , Kian-Fritz Röhrs , Jana Ackmann , Hristo Varbanov , Franziska Müller et al.
Progress in Neurobiology, 2021, 197, pp.101900. ⟨10.1016/j.pneurobio.2020.101900⟩
Journal articles hal-02940990v1

Activation chronique du récepteur de la sérotonine de type 4 : Effet préventif dans un model murin de la maladied’Alzheimer. (Conférencière invitée)

Patrizia Giannoni , Florence Gaven , Kévin Baranger , Santiago Rivera , Philippe Marin et al.
Réunion francophone sur la maladie d'Alzheimer, Jun 2014, Montpellier, France
Conference papers hal-02918585v1

Increasing spinal 5-HT 2A receptor responsiveness mediates anti-allodynic effect and potentiates fluoxetine efficacy in neuropathic rats. Evidence for GABA release

Amandine Dupuis , Anne-Sophie Wattiez , Jérémy Pinguet , Damien Richard Richard , Frédéric Libert et al.
Pharmacological Research, 2017, 118, pp.93 - 103. ⟨10.1016/j.phrs.2016.09.021⟩
Journal articles hal-01668391v1
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Classification and Signaling Characteristics of 5-HT Receptors: Towards the Concept of 5-HT Receptosomes

Philippe Marin , Carine Becamel , Séverine Chaumont-Dubel , Franck Vandermoere , Joël Bockaert et al.
Handbook of Behavioral Neuroscience, 31 (Chapter 5), pp.91-120, 2020, Handbook of Behavioral Neurobiology of Serotonin, ⟨10.1016/B978-0-444-64125-0.00005-0⟩
Book sections hal-02491823v1
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Neuronal 5-HT metabotropic receptors: fine-tuning of their structure, signaling, and roles in synaptic modulation

Joël Bockaert , Sylvie Claeysen , Carine Becamel , Aline Dumuis , Philippe Marin et al.
Cell and Tissue Research, 2006, 326 (2), pp.553-572. ⟨10.1007/s00441-006-0286-1⟩
Journal articles hal-02484323v1
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Concentrative ER export of the serotonin transporter relies exclusively on an interaction with Sec24C

Sonja Sucic , Ali El-Kasaby , Subhodeep Sarker , Harald Sitte , Philippe Marin et al.
16th Scientific Symposium of the Austrian Pharmacological Society (APHAR), Nov 2010, Vienne, Austria. pp.A11, ⟨10.1186/1471-2210-10-S1-A11⟩
Conference papers inserm-00668429v1

Physical interaction between neurofibromin and serotonin 5-HT 6 receptor promotes receptor constitutive activity

Wissem Deraredj Nadim , Séverine Chaumont-Dubel , Fahima Madouri , Laetitia Cobret , Marie-Ludivine de Tauzia et al.
Proceedings of the National Academy of Sciences of the United States of America, 2016, 113 (43), pp.12310 - 12315. ⟨10.1073/pnas.1600914113⟩
Journal articles hal-01407899v1

Deciphering beta-arrestin-dependent signaling by RPPA

Nathalie Langonné Gallay , Elisabeth Cassier , Thomas Bourquard , Christophe Gauthier , Thomas Boulo et al.
1. International Symposium of Microgenomics, May 2014, Paris, France. , 2014, 1st International Symposium of Microgenomics
Conference poster hal-02743217v1