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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
Frédéric Lassagne
,
Timothy Langlais
,
Elsa Caytan
,
Emmanuelle Limanton
,
Ludovic Paquin
et al.
Journal articles
hal-03867783v1
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Reactivity Under Microwave Irradiation of 2-amino 4H-chromene-3-carbonitrile as tool for the construction of potential bioactive derivatives
Ali Bouattour
,
Mehdi Fakhfakh
,
Houcine Ammar
,
Ludovic Paquin
,
Jean-Pierre Bazureau
et al.
3rd International Electronic Conference on Medicinal Chemistry, Nov 2022, Online, France
Conference papers
hal-03872422v1
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Eimeria tenella ROP kinase 2 induces p38 MAPK cellular pathway
Adeline Ribeiro E Silva
,
Mamadou Diallo
,
Alix Sausset
,
Thomas Robert
,
Stéphane Bach
et al.
Journées d’Animation Scientifique du Département Santé Animale (JAS SA), Oct 2022, Anglet, France.
Conference poster
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Thiazolo[5,4- f ]quinoxalines, Oxazolo[5,4- f ]quinoxalines and Pyrazino[ b,e ]isatins: Synthesis from 6-Aminoquinoxalines and Properties
Frédéric Lassagne
,
Joshua M. Sims
,
William Erb
,
Olivier Mongin
,
Nicolas Richy
et al.
Journal articles
hal-03269555v1
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Practical approach to N-benzyl derivatives of 2-amino-8-methoxy-4H-chromene-3-carbonitrile by reductive amination: Exploration of their effects against protein kinases and in silico ADME profiling
Marwa Dhiabi
,
Ali Bouattour
,
Mehdi Fakhfakh
,
Souhir Abid
,
Ludovic Paquin
et al.
Journal articles
hal-03867314v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
Camille Déliko Dago
,
Christelle Ambeu
,
Wacothon-Karime Coulibaly
,
Yves-Alain Békro
,
Janat Mamyrbékova
et al.
Journal articles
hal-01187427v1
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Discovery of simplified benzazole fragments derived from the marine benzosceptrin B as necroptosis inhibitors involving the receptor interacting protein Kinase-1
Mohamed Benchekroun
,
Ludmila Ermolenko
,
Minh Quan Tran
,
Agathe Vagneux
,
Hristo Nedev
et al.
Journal articles
hal-03004425v2
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An in silico approach for the discovery of CDK5/p25 interaction inhibitors.
Bing Zhang
,
Caroline Corbel
,
Françoise Guéritte
,
Cyril Couturier
,
Stéphane Bach
et al.
Journal articles
istex
hal-00628754v1
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Identification of intracellular targets of small molecular weight chemical compounds using affinity chromatography.
Damien Guiffant
,
Déborah Tribouillard
,
Fabienne Gug
,
Hervé Galons
,
Laurent Meijer
et al.
Journal articles
hal-00169462v1
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Synthesis and kinase inhibitory potencies of new pyrido[3,4-g]quinazolines substituted at the 8-position
Yannick Esvan
,
Béatrice Josselin
,
Blandine Baratte
,
Stéphane Bach
,
Sandrine Ruchaud
et al.
Journal articles
hal-02926291v1
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New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis
Helmi Tazarki
,
Wael Zeinyeh
,
Yannick J. Esvan
,
Stefan Knapp
,
Deep Chatterjee
et al.
Journal articles
hal-02150788v1
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Bioprospecting Marine Plankton
Heni Abida
,
Sandrine Ruchaud
,
Laurent Rios
,
Anne Humeau
,
Ian Probert
et al.
Journal articles
hal-01258229v1
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Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases
Viet Hung Dao
,
Isabelle Ourliac-Garnier
,
Cédric Logé
,
Florence Mccarthy
,
Stéphane Bach
et al.
Journal articles
hal-03428747v1
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High-Throughput Screening of marine resources
Arnaud Hochard
,
Luc Reininger
,
Sandrine Ruchaud
,
Stéphane Bach
Book sections
hal-03871307v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury Halauko
et al.
Journal articles
hal-03875302v1
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Nigratine as first-in-class dual inhibitor of necroptosis and ferroptosis regulated cell death
Claire Delehouzé
,
Arnaud Comte
,
Marcelle Hauteville
,
Peter G Goekjian
,
Marie-Thérèse Dimanche-Boitrel
et al.
2022
Preprints, Working Papers, ...
hal-03867390v1
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The Franco-Brazilian network on natural products (FB2NP): a new network promoting cooperation and exchanges in natural products research
Jackson Almeida
,
Raphaël Grougnet
,
Lucindo Quintans
,
Marc Feuilloley
,
Thomas Robert
et al.
Journal articles
hal-03592226v1
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
,
Wacothon Karime Coulibaly
,
Yves-Alain Bekro
,
Janat A. Mamyrbekova-Bekro
,
Beatrice Foll-Josselin
et al.
Journal articles
hal-01414293v1
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Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration
Viet Hung Dao
,
Isabelle Ourliac-Garnier
,
Marc-Antoine Bazin
,
Catherine Jacquot
,
Blandine Baratte
et al.
Journal articles
hal-03011408v1
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Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition
Hannah Winfield
,
Michael Cahill
,
Kevin O'Shea
,
Larry Pierce
,
Thomas Robert
et al.
Journal articles
hal-03011414v1
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Identification of potential cellular targets of aloisine A by affinity chromatography.
Caroline Corbel
,
Rose Haddoub
,
Damien Guiffant
,
Olivier Lozach
,
David Gueyrard
et al.
Journal articles
istex
hal-00416033v1
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Improved tumor control through circadian clock induction by Seliciclib, a cyclin-dependent kinase inhibitor.
Ida Iurisci
,
Elisabeth Filipski
,
Jens Reinhardt
,
Stéphane Bach
,
Athos Gianella-Borradori
et al.
Journal articles
hal-00169367v1
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Neurymenolide A, a Novel Mitotic Spindle Poison from the New Caledonian Rhodophyta Phacelocarpus neurymenioides
Sofia-Eléna Motuhi
,
Omid Feizbakhsh
,
Beatrice Foll-Josselin
,
Blandine Baratte
,
Claire Delehouze
et al.
Marine drugs, 2019, Cell Stress, Canonical and Non-Canonical Cell Death Modalities by Marine Natural Compounds and Derivatives, 17 (2), pp.93. ⟨10.3390/md17020093⟩
Journal articles
hal-02088007v1
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The Canadian Prairie Plant Thermopsis rhombifolia Contains Luteolin, a Flavone that Inhibits Cyclin Dependent Kinase 9 and Arrest Cells in the G1-Phase of the Cell Cycle
Jan Tuescher
,
Deserae Tailfeathers
,
Sophie Kernéis
,
Blandine Baratte
,
Sandrine Ruchaud
et al.
Journal articles
hal-03868334v1
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
Bruno Oyallon
,
Marie Brachet-Botineau
,
Cédric Logé
,
Pascal Bonnet
,
Mohamed Souab
et al.
Journal articles
hal-03408667v1
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Synthesis and evaluation of C3 substituted chalcone‐based derivatives of 7‐azaindole as protein kinase inhibitors
Malikotsi Qhobosheane
,
Lesetja Legoabe
,
Béatrice Josselin
,
Stéphane Bach
,
Sandrine Ruchaud
et al.
Journal articles
hal-02906292v1
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First BRET-based screening assay performed in budding yeast leads to the discovery of CDK5/p25 interaction inhibitors.
Caroline Corbel
,
Qian Wang
,
Hadjira Bousserouel
,
Amel Hamdi
,
Bing Zhang
et al.
Journal articles
istex
hal-00628746v1
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A Comparative Insight of Potassium Vanadates as Positive Electrode Materials for Li Batteries: Influence of the Long-Range and Local Structure
Rita Baddour-Hadjean
,
Arezki Boudaoud
,
Stéphane Bach
,
Nicolas Emery
,
Jean Pierre Pereira-Ramos
et al.
Journal articles
hal-03131789v1
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From benzofuro-, benzothieno- and 10-methylindolo-[2,3-b]-fused benzothiopyrano[4,3,2-de]quinolines to the corresponding benzothiopyrano[4,3,2-de]1,8-naphthyridines: synthesis and properties of these hexacyclic heteroaromatic compounds
Nicolas Mast
,
William Erb
,
Lionel Nauton
,
Pascale Moreau
,
Olivier Mongin
et al.
Journal articles
hal-03904365v1
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From simple quinoxalines to potent oxazolo[5,4- f ]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)
Frédéric Lassagne
,
Camille Duguépéroux
,
Carlos Roca
,
Concepcion Perez
,
Ana Martinez
et al.
Journal articles
hal-03011380v1
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