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authIdHal_s : stephane-l-bach
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines

Frédéric Lassagne , Timothy Langlais , Elsa Caytan , Emmanuelle Limanton , Ludovic Paquin et al.
Molecules, 2018, 23 (11), pp.2961. ⟨10.3390/molecules23112961⟩
Journal articles hal-03867783v1
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Reactivity Under Microwave Irradiation of 2-amino 4H-chromene-3-carbonitrile as tool for the construction of potential bioactive derivatives

Ali Bouattour , Mehdi Fakhfakh , Houcine Ammar , Ludovic Paquin , Jean-Pierre Bazureau et al.
3rd International Electronic Conference on Medicinal Chemistry, Nov 2022, Online, France
Conference papers hal-03872422v1

Eimeria tenella ROP kinase 2 induces p38 MAPK cellular pathway

Adeline Ribeiro E Silva , Mamadou Diallo , Alix Sausset , Thomas Robert , Stéphane Bach et al.
Journées d’Animation Scientifique du Département Santé Animale (JAS SA), Oct 2022, Anglet, France.
Conference poster hal-03852796v1
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Thiazolo[5,4- f ]quinoxalines, Oxazolo[5,4- f ]quinoxalines and Pyrazino[ b,e ]isatins: Synthesis from 6-Aminoquinoxalines and Properties

Frédéric Lassagne , Joshua M. Sims , William Erb , Olivier Mongin , Nicolas Richy et al.
European Journal of Organic Chemistry, 2021, 2021 (19), pp.2756-2763. ⟨10.1002/ejoc.202100362⟩
Journal articles hal-03269555v1
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Practical approach to N-benzyl derivatives of 2-amino-8-methoxy-4H-chromene-3-carbonitrile by reductive amination: Exploration of their effects against protein kinases and in silico ADME profiling

Marwa Dhiabi , Ali Bouattour , Mehdi Fakhfakh , Souhir Abid , Ludovic Paquin et al.
Journal of Molecular Structure, 2023, 1274 (Part 1), pp.134319. ⟨10.1016/j.molstruc.2022.134319⟩
Journal articles hal-03867314v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases

Camille Déliko Dago , Christelle Ambeu , Wacothon-Karime Coulibaly , Yves-Alain Békro , Janat Mamyrbékova et al.
Molecules, 2015, 20 (7), pp.12412-12435. ⟨10.3390/molecules200712412⟩
Journal articles hal-01187427v1
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Discovery of simplified benzazole fragments derived from the marine benzosceptrin B as necroptosis inhibitors involving the receptor interacting protein Kinase-1

Mohamed Benchekroun , Ludmila Ermolenko , Minh Quan Tran , Agathe Vagneux , Hristo Nedev et al.
European Journal of Medicinal Chemistry, 2020, 201, pp.112337. ⟨10.1016/j.ejmech.2020.112337⟩
Journal articles hal-03004425v2

An in silico approach for the discovery of CDK5/p25 interaction inhibitors.

Bing Zhang , Caroline Corbel , Françoise Guéritte , Cyril Couturier , Stéphane Bach et al.
Biotechnology Journal, 2011, 6 (7), pp.871-881. ⟨10.1002/biot.201100139⟩
Journal articles istex hal-00628754v1

Identification of intracellular targets of small molecular weight chemical compounds using affinity chromatography.

Damien Guiffant , Déborah Tribouillard , Fabienne Gug , Hervé Galons , Laurent Meijer et al.
Biotechnology Journal, 2007, 2 (1), pp.68-75. ⟨10.1002/biot.200600223⟩
Journal articles hal-00169462v1

Synthesis and kinase inhibitory potencies of new pyrido[3,4-g]quinazolines substituted at the 8-position

Yannick Esvan , Béatrice Josselin , Blandine Baratte , Stéphane Bach , Sandrine Ruchaud et al.
ARKIVOC - Online Journal of Organic Chemistry, 2020, 2020 (7), pp.105-116. ⟨10.24820/ark.5550190.p011.268⟩
Journal articles hal-02926291v1
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New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis

Helmi Tazarki , Wael Zeinyeh , Yannick J. Esvan , Stefan Knapp , Deep Chatterjee et al.
European Journal of Medicinal Chemistry, 2019, 166, pp.304-317. ⟨10.1016/j.ejmech.2019.01.052⟩
Journal articles hal-02150788v1
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Bioprospecting Marine Plankton

Heni Abida , Sandrine Ruchaud , Laurent Rios , Anne Humeau , Ian Probert et al.
Marine drugs, 2013, 11 (11), pp.4594-4611. ⟨10.3390/md11114594⟩
Journal articles hal-01258229v1
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Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases

Viet Hung Dao , Isabelle Ourliac-Garnier , Cédric Logé , Florence Mccarthy , Stéphane Bach et al.
Molecules, 2021, 26 (21), pp.6572. ⟨10.3390/molecules26216572⟩
Journal articles hal-03428747v1
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High-Throughput Screening of marine resources

Arnaud Hochard , Luc Reininger , Sandrine Ruchaud , Stéphane Bach
Outstanding Marine Molecules, 2015, ⟨10.1002/9783527681501.ch23⟩
Book sections hal-03871307v1

Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells

Madani Hedidi , Julien Maillard , William Erb , Frédéric Lassagne , Yury Halauko et al.
Tetrahedron, 2016, 72 (39), pp.6467 - 6476. ⟨10.1016/j.tet.2016.08.056⟩
Journal articles hal-03875302v1
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Nigratine as first-in-class dual inhibitor of necroptosis and ferroptosis regulated cell death

Claire Delehouzé , Arnaud Comte , Marcelle Hauteville , Peter G Goekjian , Marie-Thérèse Dimanche-Boitrel et al.
Preprints, Working Papers, ... hal-03867390v1
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The Franco-Brazilian network on natural products (FB2NP): a new network promoting cooperation and exchanges in natural products research

Jackson Almeida , Raphaël Grougnet , Lucindo Quintans , Marc Feuilloley , Thomas Robert et al.
Journal articles hal-03592226v1

Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors

Camille Déliko Dago , Wacothon Karime Coulibaly , Yves-Alain Bekro , Janat A. Mamyrbekova-Bekro , Beatrice Foll-Josselin et al.
Medicinal Chemistry Research, 2016, 25 (12), pp.2940--2958. ⟨10.1007/s00044-016-1719-3⟩
Journal articles hal-01414293v1

Benzofuro[3,2-d]pyrimidines inspired from cercosporamide CaPkc1 inhibitor: Synthesis and evaluation of fluconazole susceptibility restoration

Viet Hung Dao , Isabelle Ourliac-Garnier , Marc-Antoine Bazin , Catherine Jacquot , Blandine Baratte et al.
Bioorganic and Medicinal Chemistry, 2018, 28 (13), pp.2250-2255. ⟨10.1016/j.bmcl.2018.05.044⟩
Journal articles hal-03011408v1

Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition

Hannah Winfield , Michael Cahill , Kevin O'Shea , Larry Pierce , Thomas Robert et al.
Bioorganic and Medicinal Chemistry, 2018, 26 (14), pp.4209-4224. ⟨10.1016/j.bmc.2018.07.012⟩
Journal articles hal-03011414v1

Identification of potential cellular targets of aloisine A by affinity chromatography.

Caroline Corbel , Rose Haddoub , Damien Guiffant , Olivier Lozach , David Gueyrard et al.
Bioorganic and Medicinal Chemistry, 2009, 17 (15), pp.5572-82. ⟨10.1016/j.bmc.2009.06.024⟩
Journal articles istex hal-00416033v1

Improved tumor control through circadian clock induction by Seliciclib, a cyclin-dependent kinase inhibitor.

Ida Iurisci , Elisabeth Filipski , Jens Reinhardt , Stéphane Bach , Athos Gianella-Borradori et al.
Cancer Research, 2006, 66 (22), pp.10720-8. ⟨10.1158/0008-5472.CAN-06-2086⟩
Journal articles hal-00169367v1
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Neurymenolide A, a Novel Mitotic Spindle Poison from the New Caledonian Rhodophyta Phacelocarpus neurymenioides

Sofia-Eléna Motuhi , Omid Feizbakhsh , Beatrice Foll-Josselin , Blandine Baratte , Claire Delehouze et al.
Marine drugs, 2019, Cell Stress, Canonical and Non-Canonical Cell Death Modalities by Marine Natural Compounds and Derivatives, 17 (2), pp.93. ⟨10.3390/md17020093⟩
Journal articles hal-02088007v1

The Canadian Prairie Plant Thermopsis rhombifolia Contains Luteolin, a Flavone that Inhibits Cyclin Dependent Kinase 9 and Arrest Cells in the G1-Phase of the Cell Cycle

Jan Tuescher , Deserae Tailfeathers , Sophie Kernéis , Blandine Baratte , Sandrine Ruchaud et al.
Journal of Natural Health Product Research, 2020, 2 (2), pp.1-14. ⟨10.33211/jnhpr.12⟩
Journal articles hal-03868334v1
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors

Bruno Oyallon , Marie Brachet-Botineau , Cédric Logé , Pascal Bonnet , Mohamed Souab et al.
European Journal of Medicinal Chemistry, 2018, 154, pp.101-109. ⟨10.1016/j.ejmech.2018.04.056⟩
Journal articles hal-03408667v1

Synthesis and evaluation of C3 substituted chalcone‐based derivatives of 7‐azaindole as protein kinase inhibitors

Malikotsi Qhobosheane , Lesetja Legoabe , Béatrice Josselin , Stéphane Bach , Sandrine Ruchaud et al.
Chemical Biology and Drug Design, In press, ⟨10.1111/cbdd.13748⟩
Journal articles hal-02906292v1

First BRET-based screening assay performed in budding yeast leads to the discovery of CDK5/p25 interaction inhibitors.

Caroline Corbel , Qian Wang , Hadjira Bousserouel , Amel Hamdi , Bing Zhang et al.
Biotechnology Journal, 2011, 6 (7), pp.860-70. ⟨10.1002/biot.201100138⟩
Journal articles istex hal-00628746v1

A Comparative Insight of Potassium Vanadates as Positive Electrode Materials for Li Batteries: Influence of the Long-Range and Local Structure

Rita Baddour-Hadjean , Arezki Boudaoud , Stéphane Bach , Nicolas Emery , Jean Pierre Pereira-Ramos et al.
Inorganic Chemistry, 2014, 53 (3), pp.1764-1772. ⟨10.1021/ic402897d⟩
Journal articles hal-03131789v1
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From benzofuro-, benzothieno- and 10-methylindolo-[2,3-b]-fused benzothiopyrano[4,3,2-de]quinolines to the corresponding benzothiopyrano[4,3,2-de]1,8-naphthyridines: synthesis and properties of these hexacyclic heteroaromatic compounds

Nicolas Mast , William Erb , Lionel Nauton , Pascale Moreau , Olivier Mongin et al.
New Journal of Chemistry, 2022, 47 (1), pp.258-283. ⟨10.1039/D2NJ04567B⟩
Journal articles hal-03904365v1
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From simple quinoxalines to potent oxazolo[5,4- f ]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)

Frédéric Lassagne , Camille Duguépéroux , Carlos Roca , Concepcion Perez , Ana Martinez et al.
Organic & Biomolecular Chemistry, 2020, 18 (1), pp.154-162. ⟨10.1039/c9ob02002k⟩
Journal articles hal-03011380v1