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Structure: Internal structure identifier : 1041883

Could we expect new praziquantel derivatives ? A meta pharmacometrics/pharmacoinformatics analysis of all antischistosomal praziquantel derivatives found in the literature

V.B. Ribeiro da Silva , B. Boucherle , Jonathan El Methni , B. Hoffmann , A.L. da Silva et al.
SAR and QSAR in Environmental Research, 2019, 30 (6), pp.383 - 401
Journal articles hal-03928621v1

The advantages and challenges raised by the chemistry of aldehydic cellulose nanofibers in medicinal chemistry

Isabelle Baussanne , Julien Bras , Bastien Watbled , Martine Demeunynck
Future Medicinal Chemistry, 2018, 10 (23), pp.2679-2683. ⟨10.4155/fmc-2018-0277⟩
Journal articles hal-02326767v1

A New Anti-CXCR4 Antibody That Blocks the CXCR4/SDF-1 Axis and Mobilizes Effector Cells

M. Broussas , N. Boute , B. Akla , Sébastien Berger , C. Beau-Larvor et al.
Molecular Cancer Therapeutics, 2016, 15, pp.1890-1899. ⟨10.1158/1535-7163.MCT-16-0041⟩
Journal articles hal-01792386v1

Micro thermal energy harvester design optimization

E. Trioux , S. Monfray , Skandar Basrour
Journal of Micromechanics and Microengineering, 2017, 27 (11), pp.114001
Journal articles hal-01700995v1

Trace-driven exploration of sharing set management strategies for cache coherence in manycores

J. Dumas , E. Guthmuller , C. Fuguet Tortolero , Frédéric Pétrot
15th IEEE International New Circuits and Systems Conference (NEWCAS'17), Jun 2017, Strasbourg, France. pp.77-80
Conference papers hal-01701046v1

2-Indolylmethylenebenzofuranones as first effective inhibitors of ABCC2

Elisabeta Baiceanu , Kim-Anh Nguyen , Lucia Gonzalez-Lobato , Rachad Nasr , Hélène Baubichon-Cortay et al.
European Journal of Medicinal Chemistry, 2016, 122, pp.408 - 418. ⟨10.1016/j.ejmech.2016.06.039⟩
Journal articles hal-01683292v1

Multianalytical Study of the Binding between a Small Chiral Molecule and a DNA Aptamer: Evidence for Asymmetric Steric Effect upon 3′- versus 5′-End Sequence Modification

Lylian Challier , Rebeca Miranda-Castro , Bertrand Barbe , Claire Fave , Benoit Limoges et al.
Analytical Chemistry, 2016, 88 (23), pp.11963 - 11971. ⟨10.1021/acs.analchem.6b04046⟩
Journal articles hal-01644688v1
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Single crystals of V-amylose complexed with bicyclic organic compounds.

Cong Anh Khanh Le , Luc Choisnard , Denis Wouessidjewe , Jean-Luc Putaux
12th International IUPAC Conference on Polymer-Solvent Complexes and Intercalates (POLYSOLVAT-12), Sep 2018, 386, pp.190007, 2019, ⟨10.1021/masy.2019000007⟩
Proceedings hal-02314449v1
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FNA fluorescence reporting within silica-zirconia porous thin films

Marine Le Goas , Nina Landreau , Valérie Guieu , Corinne Ravelet , Frederic Peyrin et al.
Aptamers in Bordeaux, Jun 2016, Bordeaux, France
Conference papers cea-02349453v1

Modulators of the Efflux Pump Cdr1p of Candida albicans: Mechanisms of Action and Chemical Features

Viet-Khoa Tran-Nguyen , Rajendra Prasad , Pierre Falson , Ahcene Boumendjel
Current Medicinal Chemistry, 2017, 24 (30), pp.1 - 12. ⟨10.2174/0929867324666170523102244⟩
Journal articles hal-02329499v1
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Virtual screening against carbohydrate-binding proteins: evaluation and application to bacterial Burkholderia ambifaria lectin

Tamir Dingjan , Emilie Gillon , Anne Imberty , Serge Perez , Elizabeth Yuriev et al.
Journal of Chemical Information and Modeling, 2018, 58 (9), pp.1976-1989. ⟨10.1021/acs.jcim.8b00185⟩
Journal articles hal-02106059v1
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Enzymatically Activated Glyco-Prodrugs of Doxorubicin Synthesized by a Catalysis-Free Diels–Alder Reaction

David Bliman , Martine Demeunynck , Pierre Leblond , Samuel Meignan , Isabelle Baussane et al.
Bioconjugate Chemistry, 2018, 29 (7), pp.2370-2381. ⟨10.1021/acs.bioconjchem.8b00314⟩
Journal articles hal-02115111v1

Responses of above- and below-ground fungal symbionts to cessation of mowing in subalpine grassland

Marie-Noëlle Binet , Diederik van Tuinen , Florence Souard , Lucile Sage , Sophie Perigon et al.
Fungal Ecology, 2017, 25, pp.14-21. ⟨10.1016/j.funeco.2016.10.001⟩
Journal articles hal-01605015v1

Specific and spatial labeling of choline-containing teichoic acids in Streptococcus pneumoniae by click chemistry

Julie Bonnet , Anne-Marie Di Guilmi , Stefan Peiβert , Claire Durmort , Benoit Gallet et al.
Chemical Communications, 2017, 53 (76), pp.10572 - 10575. ⟨10.1039/c7cc05646j⟩
Journal articles hal-01613804v1

Disruption of Fibers from the Tau Model AcPHF6 by Naturally Occurring Aurones and Synthetic Analogues

Laurent Lunven , Hugues Bonnet , Samir Yahiaoui , Wei Yi , Laurène da Costa et al.
ACS Chemical Neuroscience, 2016, 7 (7), pp.995 - 1003. ⟨10.1021/acschemneuro.6b00102⟩
Journal articles hal-01644834v1

Efficient functional neutralization of lethal peptide toxins in vivo by oligonucleotides

Tarek Mohamed Abd El-Aziz , Corinne Ravelet , Jordi Molgó , Emmanuelle Fiore , Simon Pale et al.
Scientific Reports, 2017, 7 (1), ⟨10.1038/s41598-017-07554-5⟩
Journal articles hal-01639599v1

Investigating the toxic effects induced by iron oxide nanoparticles on neuroblastoma cell line: an integrative study combining cytotoxic, genotoxic and proteomic tools

Dalel Askri , Valérie Cunin , David Béal , Sylvie Berthier , Benoit Chovelon et al.
Nanotoxicology, 2019, pp.1-20. ⟨10.1080/17435390.2019.1621399⟩
Journal articles hal-02189282v1

Evaluation of a Computed Assisted Medical Intervention (CAMI) systems in scientific autopsy

F. Grenier , Sandrine Voros , V. Scolan , F. Paysant , J. Boutonnat et al.
Journal of Forensic Radiology and Imaging, 2017, 11, pp.6 - 11. ⟨10.1016/j.jofri.2017.08.006⟩
Journal articles hal-01668727v1
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Synthesis and biological evaluation of novel imidazolinic, thiazolinic derivatives and aminosugars

Vinicius Barros Ribeiro Da Silva
Agricultural sciences. Universidade federal de Pernambuco (Récife, Brésil), 2017. Portuguese. ⟨NNT : 2017GREAV022⟩
Theses tel-01684234v1
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Synthèse de nouveaux analogues de nucléosides potentiellement antiviraux.

Flavia Cristina Rosa Alvarenga
Médecine humaine et pathologie. Université Grenoble Alpes, 2016. Français. ⟨NNT : 2016GREAV068⟩
Theses tel-02003332v1
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Synthesis of a poison frog bioactive alkaloids

Sara Mazeh
Organic chemistry. Université Grenoble Alpes, 2019. English. ⟨NNT : 2019GREAV043⟩
Theses tel-02613846v1

Selective luminescentes Étiquetage de l'ADN et de l'ARN quadruplex par tc-Extended ruthénium Light-Up Sondes.

D. Saadallah , M. Bellakhal , S. Amor , J.-F. Lefebvre , M. Chavarot-Kerlidou et al.
Chemistry , 2017, 23 (21), pp.4967-4972. ⟨10.1002/chem.201605948⟩
Journal articles hal-01482247v1
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Exploring the structure-activity relationship of benzylidene-2,3-dihydro-1H-inden-1-one compared to benzofuran-3(2H)-one derivatives as inhibitors of tau amyloid fibers

Emeline Boukherrouba , Camille Larosa , Kim-Anh Nguyen , Jérémy Caburet , Laurent Lunven et al.
European Journal of Medicinal Chemistry, 2022, 231, pp.114139. ⟨10.1016/j.ejmech.2022.114139⟩
Journal articles hal-04014492v1
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Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2

Emile Roussel , Viet-Khoa Tran-Nguyen , Khalid Bouhedjar , Mohamed Abdesselem Dems , Amine Belaidi et al.
European Journal of Medicinal Chemistry, 2019, 184, pp.111772. ⟨10.1016/j.ejmech.2019.111772⟩
Journal articles hal-02442448v1

Nascent teichoic acids insertion into the cell wall directs the localization and activity of the major pneumococcal autolysin LytA

Julie Bonnet , Claire Durmort , I. Mortier-Barrière , N. Campo , M. Jacq et al.
The Cell Surface, 2018, 2, pp.24 - 37. ⟨10.1016/j.tcsw.2018.05.001⟩
Journal articles hal-01823775v1

Miscellaneous nanoaggregates made of β-CD esters synthesised by an enzymatic pathway

L. Choisnard , A. Geze , B.G.J. Yameogo , J.L. Putaux , D. Wouessidjewe et al.
International Journal of Pharmaceutics, 2007, 344 (1-2), pp.26-32. ⟨10.1016/j.ijpharm.2007.06.026⟩
Journal articles istex hal-00305547v1

Leurre GD-FXa mutant

Aline Thomas , Raphaël Marlu , Benoit Polack , Atanur Ersayin , Marie Claire Dagher et al.
France, Patent n° : FR1753060. 2017
Patents hal-03068391v1
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Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens

Hamza Olleik , Samir Yahiaoui , Brayan Roulier , Elise Courvoisier-Dezord , Josette Perrier et al.
European Journal of Medicinal Chemistry, 2019, 165, pp.133-141. ⟨10.1016/j.ejmech.2019.01.022⟩
Journal articles hal-01988325v1

A ππ* State Enables Photoaccumulation of Charges on a π‑Extended Dipyridophenazine Ligand in a Ru(II) Polypyridine Complex

Julian Schindler , Ying Zhang , Philipp Traber , Lefebvre Jean-François , Stephan Kupfer et al.
Journal of Physical Chemistry C, 2018, 122 (1), pp.83-95. ⟨10.1021/acs.jpcc.7b08989⟩
Journal articles hal-01775421v1

Enzymatically Activated Glyco-Prodrugs of Doxorubicin Synthesized by a Catalysis-Free Diels−Alder Reaction

David Bliman , Martine Demeunynck , Pierre Leblond , Samuel Meignan , Sébastien Fort et al.
Bioconjugate Chemistry, 2018
Journal articles hal-03773343v1