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Structure: Internal structure identifier : 207869

Substituted thiazolamide coupled to a redox delivery system: a new γ-secretase inhibitor with enhanced pharmacokinetic profile

Younes Laras , Gilles Quéléver , Cédrik Garino , Nicolas Pietrancosta , Mahmoud Sheha et al.
Organic & Biomolecular Chemistry, 2005, 3 (4), pp.612-618. ⟨10.1039/b415090b⟩
Journal articles istex hal-02351730v1

Development of a L-Tryptophan-Based Ligand for Regioselective Copper Catalyzed N 2 -Arylation of 1,2,3-Triazoles

Alexandra Basilio Lopes , Patrick Wagner , Arthur Eugen Kümmerle , Frédéric Bihel , Jean-Jacques Bourguignon et al.
ChemistrySelect, 2017, 2 (22), pp.6544-6548. ⟨10.1002/slct.201701498⟩
Journal articles hal-02368798v1
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Stratégies de synthèse d’un nouvel antipsychotique potentiel : cascades réactionnelles palladocatalysées : un outil puissant pour la synthèse de structures polycycliques complexes et hautement fonctionnalisées

Jessie Joussot
Autre. Université de Strasbourg, 2015. Français. ⟨NNT : 2015STRAF016⟩
Theses tel-01255212v1
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New Culture Media for Fast, Sensitive and User-Friendly Detection of E.Coli and/or Coliform Bacteria

Etienne Schaeffer , Jacques Haiech , Jean-Luc Galzi
Research & Reviews: Journal of Microbiology and Biotechnology, 2017, 6 (3), pp.50-61
Journal articles hal-02191030v1
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An Antedrug of the CXCL12 Neutraligand Blocks Experimental Allergic Asthma without Systemic Effect in Mice

Francois Daubeuf , Muriel Hachet-Haas , Patrick Gizzi , Vincent Gasparik , Dominique Bonnet et al.
Journal of Biological Chemistry, 2013, 288 (17), pp.11865-11876. ⟨10.1074/jbc.M112.449348⟩
Journal articles hal-02194500v1
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QSPR modelling -a valuable support in HTS quality control

Fiorella Ruggiu , Patrick Gizzi , Jean-Luc Galzi , Marcel Hibert , Jacques Haiech et al.
Analytical Chemistry, 2014, ⟨10.1021/ac403544k⟩
Journal articles hal-02196042v1
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Parcourir l’histoire de l’intelligence artificielle, pour mieux la définir et la comprendre

Jacques Haiech
médecine/sciences, 2020, 36 (10), pp.919-923. ⟨10.1051/medsci/2020145⟩
Journal articles hal-02960791v1

Synthesis and biological properties of conjugates between fluoroquinolones and a N3′′-functionalized pyochelin

Sabrina Noël , Veronique Gasser , Bénédicte Pesset , Francoise Hoegy , Didier Rognan et al.
Organic & Biomolecular Chemistry, 2011, 9 (24), pp.8288. ⟨10.1039/c1ob06250f⟩
Journal articles hal-02988912v1

A Summer School for Structuring the Chemoinformatics Community

Didier Rognan , Alexandre Varnek
Molecular Informatics, 2014, 33 (6-7), pp.390-390. ⟨10.1002/minf.201480631⟩
Journal articles hal-03150639v1

Development of a Peptidomimetic Antagonist of Neuropeptide FF Receptors for the Prevention of Opioid-Induced Hyperalgesia

Frédéric Bihel , Jean-Paul Humbert , Severine Schneider , Isabelle Bertin , Patrick Wagner et al.
ACS Chemical Neuroscience, 2015, 6 (3), pp.438-445. ⟨10.1021/cn500219h⟩
Journal articles hal-03198603v1

Predicting Ligand Binding Modes from Neural Networks Trained on Protein–Ligand Interaction Fingerprints

Vladimir Chupakhin , Gilles Marcou , Igor Baskin , Alexandre Varnek , Didier Rognan et al.
Journal of Chemical Information and Modeling, 2013, 53 (4), pp.763-772. ⟨10.1021/ci300200r⟩
Journal articles hal-03142314v1
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Modeling of CCR5 Recognition by HIV-1 gp120: How the Viral Protein Exploits the Conformational Plasticity of the Coreceptor

Célien Jacquemard , Florian Koensgen , Philippe Colin , Bernard Lagane , Esther Kellenberger et al.
Viruses, 2021, 13 (7), pp.1395. ⟨10.3390/v13071395⟩
Journal articles hal-03320721v1
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The human pre-replication complex is an open complex

Jian Li , Jiangqing Dong , Weitao Wang , Daqi Yu , Xinyu Fan et al.
Cell, 2023, 186 (1), pp.98-111.e21. ⟨10.1016/j.cell.2022.12.008⟩
Journal articles hal-03974204v1

Prendre la mesure d’une culture ouverte et responsable

Claire Marris , Thomas Heams , Francois Kepes , Luis Campos , Pierre Monsan et al.
3. Colloque Sciences de la vie en société, Dec 2012, Paris, France
Conference papers hal-01628091v1

Recent advances in the biology and chemistry of the flavaglines

Nigel Ribeiro , Frédéric Thuaud , Canan G Nebigil , Laurent Désaubry
Bioorganic and Medicinal Chemistry Letters, 2012, 20 (6), pp.1857-1864. ⟨10.1016/j.bmc.2011.10.048⟩
Journal articles hal-02391066v1
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Lithium reverses mechanical allodynia through a mu opioid-dependent mechanism

Ivan Weinsanto , Jinane Mouheiche , Alexis Laux-Biehlmann , Maya Aouad , Tando Maduna et al.
Molecular Pain, 2018, 14, pp.174480691775414. ⟨10.1177/1744806917754142⟩
Journal articles hal-02061235v1
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Synthèse d'agonistes non-peptidiques du récepteur à la prokinéticine PKR1

Marine Charavin
Chimie thérapeutique. Université de Strasbourg, 2014. Français. ⟨NNT : 2014STRAF047⟩
Theses tel-02003517v1
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Conception et caractérisation d'antagonistes allostériques de l'intégrine α5β1 pour le traitement des glioblastomes

Anne-Marie Ray
Sciences agricoles. Université de Strasbourg, 2013. Français. ⟨NNT : 2013STRAF032⟩
Theses tel-02003521v1
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Erratum to: "CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

Saleh Mones , Burkhard Gess , Benoit Bordignon , Alexandre Altie , Peter Young et al.
Orphanet Journal of Rare Diseases, 2016, 11, ⟨10.1186/s13023-015-0354-2⟩
Journal articles hal-02630248v1

Expeditious Syntheses of (±)- allo -Sedamine and (±)- allo -Lobeline via a Combination of Aza-Sakurai-Hosomi and Hydroformylation Reactions

Thomas Spangenberg , Etienne Airiau , Mathieu Thuong , Morgan Donnard , Manuella Billet et al.
SYNLETT, 2008, 2008 (18), pp.2859-2863. ⟨10.1055/s-0028-1083543⟩
Journal articles hal-02105037v1
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Human erythrocytes release ATP by a novel pathway involving VDAC oligomerization independent of pannexin-1

Irene Marginedas-Freixa , Cora Lilia Alvarez , Martina Moras , María Florencia Leal Denis , Claude Hattab et al.
Scientific Reports, 2018, 8, pp.11384. ⟨10.1038/s41598-018-29885-7⟩
Journal articles hal-02368694v1
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Activating the apelin receptor with LIT01-196, a metabolically stable apelin analog, reverses AVP-induced antidiuresis and hyponatremia

Adrien Flahault , Pierre-Emmanuel Girault-Sotias , Mathilde Keck , Rodrigo Alvear-Perez , Nadia de Mota et al.
Nature Communications, 2021, 12 (1), ⟨10.1038/s41467-020-20560-y⟩
Journal articles hal-03285794v1

Bioisosteric modification of flavaglines

Qian Zhao , Annemilaï Tijeras-Raballand , Armand de Gramont , Eric Raymond , Laurent Désaubry et al.
Tetrahedron Letters, 2016, 57 (26), pp.2943-2944. ⟨10.1016/j.tetlet.2016.05.089⟩
Journal articles hal-03533709v1

Etude de l’activité anti-tumorale de nouveaux ligands ciblant LINGO-1 pour le traitement des glioblastomes

Wanyin Chen , Anthony Guillemain , Lauren Blot , Fabienne Fasani , Esther Kellenberger et al.
Colloque de l’ADOC, Jul 2019, Orléans, France
Conference poster hal-03686230v1
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Three Cheers for Nitrogen: Aza-DKPs, the Aza Analogues of 2,5-Diketopiperazines

Timothé Maujean , Nicolas Girard , A. Ganesan , Mihaela Gulea , Dominique Bonnet et al.
RSC Advances, 2020, 10 (71), pp.43358-43370. ⟨10.1039/d0ra09457a⟩
Journal articles hal-03441420v1
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Targeting the Central Pocket of the Pseudomonas aeruginosa lectin LecA

Eike Siebs , Elena Shanina , Sakonwan Kuhaudomlarp , Priscila da Silva Figueiredo Celestino Gomes , Cloé Fortin et al.
ChemBioChem, 2021, ⟨10.1002/cbic.202100563⟩
Journal articles hal-03438182v1
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The mTOR-S6 kinase pathway promotes stress granule assembly

Aristeidis Sfakianos , Laura Mellor , Yoke Fei Pang , Paraskevi Kritsiligkou , Hope Needs et al.
Cell Death and Differentiation, 2018, 25 (10), pp.1766-1780. ⟨10.1038/s41418-018-0076-9⟩
Journal articles hal-02361603v1
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Antiallodynic action of phosphodiesterase inhibitors in a mouse model of peripheral nerve injury

Salim Megat , Sylvain Hugel , Sarah Journée , Yohann Bohren , Adrien Lacaud et al.
Neuropharmacology, 2022, 205, pp.108909. ⟨10.1016/j.neuropharm.2021.108909⟩
Journal articles hal-03842284v1
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Molecular Diversity of Cyclooctatetraenes through Palladium-Catalyzed Cascade Reactions

Sarah Blouin , Romain Pertschi , Angèle Schoenfelder , Jean Suffert , Gaëlle Blond et al.
Advanced Synthesis and Catalysis, 2018, 360 (11), pp.2166-2171. ⟨10.1002/adsc.201800110⟩
Journal articles hal-02322480v1
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LIT-PCBA: An Unbiased Dataset for Machine Learning and Virtual Screening

Viet-Khoa Tran-Nguyen , Célien Jacquemard , Didier Rognan
Journal of Chemical Information and Modeling, 2020, 60 (9), pp.4263-4273. ⟨10.1021/acs.jcim.0c00155⟩
Journal articles hal-03013622v1