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Substituted thiazolamide coupled to a redox delivery system: a new γ-secretase inhibitor with enhanced pharmacokinetic profile
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Cédrik Garino
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istex
hal-02351730v1
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Development of a L-Tryptophan-Based Ligand for Regioselective Copper Catalyzed N 2 -Arylation of 1,2,3-Triazoles
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Patrick Wagner
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hal-02368798v1
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Stratégies de synthèse d’un nouvel antipsychotique potentiel : cascades réactionnelles palladocatalysées : un outil puissant pour la synthèse de structures polycycliques complexes et hautement fonctionnalisées
Jessie Joussot
Theses
tel-01255212v1
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New Culture Media for Fast, Sensitive and User-Friendly Detection of E.Coli and/or Coliform Bacteria
Etienne Schaeffer
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Jacques Haiech
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Jean-Luc Galzi
Research & Reviews: Journal of Microbiology and Biotechnology, 2017, 6 (3), pp.50-61
Journal articles
hal-02191030v1
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An Antedrug of the CXCL12 Neutraligand Blocks Experimental Allergic Asthma without Systemic Effect in Mice
Francois Daubeuf
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QSPR modelling -a valuable support in HTS quality control
Fiorella Ruggiu
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Patrick Gizzi
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Parcourir l’histoire de l’intelligence artificielle, pour mieux la définir et la comprendre
Jacques Haiech
Journal articles
hal-02960791v1
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Synthesis and biological properties of conjugates between fluoroquinolones and a N3′′-functionalized pyochelin
Sabrina Noël
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Veronique Gasser
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A Summer School for Structuring the Chemoinformatics Community
Didier Rognan
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Alexandre Varnek
Journal articles
hal-03150639v1
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Development of a Peptidomimetic Antagonist of Neuropeptide FF Receptors for the Prevention of Opioid-Induced Hyperalgesia
Frédéric Bihel
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Jean-Paul Humbert
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Severine Schneider
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Isabelle Bertin
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Patrick Wagner
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hal-03198603v1
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Predicting Ligand Binding Modes from Neural Networks Trained on Protein–Ligand Interaction Fingerprints
Vladimir Chupakhin
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Gilles Marcou
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Igor Baskin
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Alexandre Varnek
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Didier Rognan
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hal-03142314v1
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Modeling of CCR5 Recognition by HIV-1 gp120: How the Viral Protein Exploits the Conformational Plasticity of the Coreceptor
Célien Jacquemard
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Bernard Lagane
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hal-03320721v1
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The human pre-replication complex is an open complex
Jian Li
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Jiangqing Dong
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Weitao Wang
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Daqi Yu
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hal-03974204v1
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Prendre la mesure d’une culture ouverte et responsable
Claire Marris
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Thomas Heams
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Francois Kepes
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Luis Campos
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Pierre Monsan
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3. Colloque Sciences de la vie en société, Dec 2012, Paris, France
Conference papers
hal-01628091v1
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Recent advances in the biology and chemistry of the flavaglines
Nigel Ribeiro
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Frédéric Thuaud
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Canan G Nebigil
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hal-02391066v1
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Lithium reverses mechanical allodynia through a mu opioid-dependent mechanism
Ivan Weinsanto
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Jinane Mouheiche
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hal-02061235v1
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Synthèse d'agonistes non-peptidiques du récepteur à la prokinéticine PKR1
Marine Charavin
Theses
tel-02003517v1
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Conception et caractérisation d'antagonistes allostériques de l'intégrine α5β1 pour le traitement des glioblastomes
Anne-Marie Ray
Theses
tel-02003521v1
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Erratum to: "CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors
Saleh Mones
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Burkhard Gess
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Benoit Bordignon
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Alexandre Altie
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Peter Young
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Journal articles
hal-02630248v1
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Expeditious Syntheses of (±)- allo -Sedamine and (±)- allo -Lobeline via a Combination of Aza-Sakurai-Hosomi and Hydroformylation Reactions
Thomas Spangenberg
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Etienne Airiau
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Mathieu Thuong
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Morgan Donnard
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Manuella Billet
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hal-02105037v1
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Human erythrocytes release ATP by a novel pathway involving VDAC oligomerization independent of pannexin-1
Irene Marginedas-Freixa
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Cora Lilia Alvarez
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Martina Moras
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María Florencia Leal Denis
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Claude Hattab
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hal-02368694v1
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Activating the apelin receptor with LIT01-196, a metabolically stable apelin analog, reverses AVP-induced antidiuresis and hyponatremia
Adrien Flahault
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Pierre-Emmanuel Girault-Sotias
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Mathilde Keck
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Rodrigo Alvear-Perez
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Nadia de Mota
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hal-03285794v1
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Bioisosteric modification of flavaglines
Qian Zhao
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Annemilaï Tijeras-Raballand
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Armand de Gramont
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hal-03533709v1
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Etude de l’activité anti-tumorale de nouveaux ligands ciblant LINGO-1 pour le traitement des glioblastomes
Wanyin Chen
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Anthony Guillemain
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Lauren Blot
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Fabienne Fasani
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Esther Kellenberger
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Colloque de l’ADOC, Jul 2019, Orléans, France
Conference poster
hal-03686230v1
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Three Cheers for Nitrogen: Aza-DKPs, the Aza Analogues of 2,5-Diketopiperazines
Timothé Maujean
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Nicolas Girard
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A. Ganesan
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Mihaela Gulea
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Dominique Bonnet
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hal-03441420v1
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Targeting the Central Pocket of the Pseudomonas aeruginosa lectin LecA
Eike Siebs
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Elena Shanina
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Sakonwan Kuhaudomlarp
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Priscila da Silva Figueiredo Celestino Gomes
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Cloé Fortin
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hal-03438182v1
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The mTOR-S6 kinase pathway promotes stress granule assembly
Aristeidis Sfakianos
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Laura Mellor
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Yoke Fei Pang
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Paraskevi Kritsiligkou
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Hope Needs
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hal-02361603v1
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Antiallodynic action of phosphodiesterase inhibitors in a mouse model of peripheral nerve injury
Salim Megat
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Sylvain Hugel
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Sarah Journée
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Yohann Bohren
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Adrien Lacaud
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hal-03842284v1
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Molecular Diversity of Cyclooctatetraenes through Palladium-Catalyzed Cascade Reactions
Sarah Blouin
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Romain Pertschi
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Angèle Schoenfelder
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Jean Suffert
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Gaëlle Blond
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Journal articles
hal-02322480v1
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LIT-PCBA: An Unbiased Dataset for Machine Learning and Virtual Screening
Viet-Khoa Tran-Nguyen
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Célien Jacquemard
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Didier Rognan
Journal articles
hal-03013622v1
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